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6-(2-fluoro-4-methoxyphenyl)-N-(3-hydroxypropyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(2S,4R)-N-ethyl-1-(2-methoxyacetyl)-4-[3-(4-methyl-1H-pyrazol-1-yl)propanamido]pyrrolidine-2-carboxamide
N-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]-2-(2,4-dioxoimidazolidin-1-yl)acetamide
(3R,4R)-3-cyclobutyl-1-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-4-methylpyrrolidin-3-ol
N-{1-[1-(adamantan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
5-methoxy-3-methyl-2-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}-1H-indole
1-[(4-methyl-1,4-oxazepan-6-yl)methyl]-3-(naphthalen-1-yl)urea
N-ethyl-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-(propan-2-yl)acetamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylpropyl)acetamide
N-benzyl-3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-N-methylpropanamide
3-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(2-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}ethyl)morpholine
2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-6-methylpyridine-3-carbonitrile
4-(1-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
N-(1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-1-oxopropan-2-yl)methanesulfonamide
3-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-[3-(methylsulfamoyl)phenyl]urea
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(2R)-1-hydroxypropan-2-yl]-5-methoxybenzamide
5-amino-N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-1H-pyrazole-3-carboxamide
4-benzyl-1-[(3,4-dihydroxyphenyl)methyl]-3-ethyl-1,4-diazepan-5-one
3-cyclopropaneamido-N,4-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]benzamide
(3S,4R)-1-(2,3-difluoro-6-methoxybenzoyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
4-[(2,6-dichloro-3-hydroxyphenyl)methyl]-1-methylpiperazine-2-carboxylic acid
methyl 3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propanoate
N-(propan-2-yl)-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
1-{1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-(5-amino-1,3,4-thiadiazol-2-yl)-1-{2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}ethan-1-one
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl]propanoic acid
3-(5-{2,7-diazaspiro[4.5]decan-2-ylmethyl}thiophen-3-yl)prop-2-yn-1-ol
3-{[3-(methoxymethyl)piperidin-1-yl]methyl}benzoic acid
1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-N-(1H-1,2,4-triazol-3-ylmethyl)piperidine-3-carboxamide
2-(2-chlorophenyl)-N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-2-hydroxyacetamide
1-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
8-[(2-methylnaphthalen-1-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
2-(adamantan-1-yl)-N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]acetamide
(3S,4R)-1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
ethyl 1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(2-phenylethyl)piperidine-4-carboxylate
1-({[4-(furan-2-yl)phenyl]carbamoyl}amino)-N-methylcyclohexane-1-carboxamide
(3S,4R)-4-(3-methoxyphenyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidine-3-carboxylic acid
4-methyl-N-(2-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-yl}ethyl)-1,2,3-thiadiazole-5-carboxamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine-4-carboxamide
methyl 2-[(4-methylphenyl)sulfamoyl]-6-(4,4,4-trifluorobutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(pyridin-3-ylformamido)ethyl]propanamide
ethyl 3-[(4-fluorophenyl)methyl]-1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidine-3-carboxylate
1-(5-chloropyridin-2-yl)-4-(2-methyl-1-benzofuran-7-carbonyl)piperazine
(2R,6R)-1-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
ethyl 1-[(4-methoxyphenyl)methyl]-5-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(phenylamino)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]pyrimidine-5-carboxamide
(1r,4r)-4-({[6-(thiophen-3-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}amino)cyclohexan-1-ol
8-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-(2-phenylethyl)piperidine-3-carboxamide