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(2S)-2-[2-(adamantan-1-yl)acetamido]pentanedioic acid
1-[2-(ethylamino)pyrimidine-5-carbonyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-(2-methylphenoxy)-1-(1,3-thiazole-4-carbonyl)piperidine-4-carboxylic acid
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-(2,2,2-trifluoroethyl)piperidine-3-carboxamide
1-(2-chlorophenyl)-3-{1-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]thiophene-3-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]propanamide
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
7-(2-methoxyethyl)-2-(4-methyl-1,3-thiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(3R,4R)-1-[(5-cyclopentylthiophen-2-yl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
6-[4-(furan-2-yl)benzoyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
1-benzyl-2-methyl-5-(2-methylpropanamido)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
7-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]-2-ethyl-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
5-(3-fluorophenoxymethyl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-pyrazole-3-carboxamide
(2S,4R)-1-[(2-aminopyridin-3-yl)methyl]-N-ethyl-4-[2-(propan-2-yloxy)acetamido]pyrrolidine-2-carboxamide
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-(pyrrolidine-1-carbonyl)pyridine
4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-1-(2,5-dihydro-1H-pyrrole-2-carbonyl)piperidine
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-benzofuran-2-carboxamide
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-[6-(methoxymethyl)pyrimidin-4-yl]-8-azabicyclo[3.2.1]octane
1-[2-({[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]imidazolidin-2-one
N-cyclohexyl-N-(pyridin-3-ylmethyl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
(1S,5R)-3-benzyl-6-[3-(1H-pyrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
4-[4-(2-methylphenyl)-1H-imidazol-2-yl]-1-(2-methylpropyl)pyrrolidin-2-one
1-{5-[(6-chloropyridazin-3-yl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-ol
6-(benzyloxy)-1-cyclohexyl-4-(2-methylpyridine-3-carbonyl)-1,4-diazepan-2-one
(3S,4R)-1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
(3aR,6aR)-2-acetyl-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[(4-chlorophenyl)methyl]-3-[(1R,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propanamide
4-(4-{[ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenyl)-2-methylbut-3-yn-2-ol
3-{[(2R)-2-hydroxypropyl]sulfamoyl}-N-[3-(pyridin-2-yl)propyl]benzamide
N-(naphthalen-1-yl)-2,8-diazaspiro[4.5]decane-2-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-N,N-dimethyl-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-sulfonamide
[(3-{[1-(furan-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
5-[3-(4-fluorophenoxymethyl)-1-(2-hydroxybutyl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
ethyl({[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl})methylamine
(dicyclopropylmethyl)({[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
(1R,5S)-3-[2-(1,2-benzoxazol-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{5-[6-amino-5-cyano-4-(3-hydroxyphenyl)pyridin-2-yl]thiophen-3-yl}acetic acid
2-methyl-7-[6-(propan-2-yl)pyrimidin-4-yl]-2,7-diazaspiro[4.4]nonane
(1S,5R)-6-(cyclopropylmethyl)-3-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 5-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-[(2E)-3-(1H-imidazol-4-yl)prop-2-enoyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(2-phenylethyl)piperidin-4-ol
2-(3-chloro-4-hydroxyphenyl)-1-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]ethan-1-one
4-[3-(2-methoxyphenoxy)azetidin-1-yl]pyridine
2-(3-methylphenyl)-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]benzamide
N-methyl-4-[3-(pyridine-2-carbonyl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
methyl 3-(2-fluorobenzamido)-5-{[(5-methylthiophen-2-yl)formamido]methyl}benzoate