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3-[5-({[1-(cyclohexylmethyl)piperidin-3-yl]amino}methyl)thiophen-2-yl]prop-2-yn-1-ol
N-benzyl-5-[4-(4-methylphenyl)piperazine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
3,4-dimethoxy-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}benzamide
2-(2-methoxyethyl)-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-1,3-benzoxazole-6-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
5-(2,5-dimethylphenoxymethyl)-N-[5-(morpholin-4-yl)pentyl]-1,2-oxazole-3-carboxamide
4-{4-[(4-tert-butylphenyl)methyl]piperazin-1-yl}-6-methoxypyrimidin-2-amine
4-{2-methyl-6-[1-(pyrimidin-2-ylmethyl)piperidin-4-yl]pyrimidin-4-yl}morpholine
5-[3-(1H-pyrazol-3-yl)phenyl]-2-(pyridin-3-yl)-1,3-benzoxazole
N-methyl-4-{[3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-N-phenylaniline
(3R,4R)-4-cyclopropyl-4-hydroxy-3-methyl-N-(naphthalen-2-yl)piperidine-1-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]acetamide
3-[({2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)methyl]-7-fluoro-1,2-dihydroquinolin-2-one
(2R)-2-amino-N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,4-dimethylpentanamide
(2S,4S)-4-amino-1-(5-ethylthiophene-3-carbonyl)-N-methylpyrrolidine-2-carboxamide
1-(diethylamino)-3-{5-[(2,2-dimethylmorpholin-4-yl)methyl]-2-methoxyphenoxy}propan-2-ol
4-ethyl-3-{1-[2-(3-hydroxyadamantan-1-yl)acetyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(dimethylamino)ethyl]-3-{5-ethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-[(2R,3R)-1'-(4-ethenylbenzoyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
4-{1-[(4-methoxypiperidin-1-yl)sulfonyl]piperidin-3-yl}benzoic acid
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
(2R)-2-hydroxy-1-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]-2-(naphthalen-2-yl)ethan-1-one
5-ethyl-2,3-dimethyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-[(4-chlorophenyl)methyl]-5-[(2R,6S)-2,6-dimethylmorpholin-4-yl]azepan-2-one
7-fluoro-2-(2-methoxyphenyl)-3-(morpholin-4-ylmethyl)quinoline
[2-(diethylamino)ethyl](ethyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-(pyridin-3-yl)-5-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}pyrimidine
(3aR,6aR)-2-cyclopentanecarbonyl-5-(3-methylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(1-methyl-1H-pyrrol-3-yl)-1-{4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
1-{4-[6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,4-diazepan-1-yl}ethan-1-one
N-[(3R,4S)-4-cyclopropyl-1-[(methylcarbamoyl)methyl]pyrrolidin-3-yl]-2-methyl-1,3-thiazole-4-carboxamide
1'-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-({1-[(2-butyl-1H-imidazol-4-yl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
(4aS,8aS)-4a-hydroxy-N-[3-(2-methoxyacetamido)phenyl]-decahydroisoquinoline-2-carboxamide
3-[5-(methanesulfonylmethyl)pyridin-2-yl]-N,N-dimethylaniline
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
9-(1,3-thiazol-2-yl)-2H,3H,4H,6H,7H,8H,9H-[1,4]oxazino[2,3-g]quinoline-3,7-dione
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-3,5-dimethyl-1,2-oxazole-4-carboxamide
N-cyclopentyl-3-{[(2,5-dimethoxyphenyl)methyl]amino}-5-(phenylsulfamoyl)benzamide
N-{2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-oxoethyl}acetamide
methyl[(3-{2-[1-(5-methylthiophene-2-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl](quinolin-8-ylmethyl)amine
2-methoxy-5-{[4-(2-methylpropyl)-1,4-diazepan-1-yl]methyl}phenol
1-(2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(4-chlorophenyl)methyl]-N-(2-cyclopentylethyl)-6-oxopiperidine-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-1-methylpiperidine-2-carboxamide
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-yl}piperidine
(2S,4R)-4-amino-1-[(5-tert-butyl-2-hydroxyphenyl)methyl]-N-ethylpyrrolidine-2-carboxamide
methyl 5-{[(3,5-dimethoxyphenyl)methyl]amino}-3-acetamido-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(4aS,7aR)-1-(2-cyclopentylacetyl)-4-[2-(dimethylamino)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-1-methyl-1H-pyrazole-3-carboxamide