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2-(3-methyl-1,2-oxazol-5-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(2R,6R)-10-methoxy-4-methyl-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[(3-tert-butyl-1,2,4-oxadiazol-5-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-{[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]methyl}thiophene-2-carboxylic acid
2-(cyclopent-1-en-1-yl)-1-(6-hydroxy-4-{[5-(hydroxymethyl)furan-2-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pentan-1-one
methyl 4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2,4-oxadiazol-3-yl]benzoate
3-{2-azaspiro[4.4]nonane-2-carbonyl}-N-(oxolan-3-ylmethyl)benzene-1-sulfonamide
4-(cyclopropylamino)-N,N-diethyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
4-{2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl}-4-oxobutane-1-sulfonamide
N-[(2-fluorophenyl)methyl]-5-(4-formyl-1,4-diazepan-1-yl)-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(4aS,8aR)-6-(1,3-benzothiazol-2-ylmethyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
4-[2-amino-3-cyano-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridin-4-yl]benzoic acid
(2S,4R)-4-amino-N-methyl-1-[3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propanoyl]pyrrolidine-2-carboxamide
2-(3-chloro-4-hydroxyphenyl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}acetamide
3-{[benzyl(methyl)amino]methyl}-1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxypiperidin-2-one
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl){[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-2-[(4-methyl-1,2,5-oxadiazol-3-yl)formamido]acetamide
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-(2-{2-amino-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindol-1-one
2-(2-chlorophenyl)-N,N,3-trimethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-methoxy-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidin-2-amine
1-[3-(3-chlorophenyl)pyrrolidin-1-yl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-3-(1H-pyrazol-4-yl)propan-1-one
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1,3-thiazol-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(cyclopropylmethyl)-1-(1H-imidazol-2-ylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(2-methyl-1H-imidazol-1-yl)propanamide
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-1-methyl-1H-imidazole-4-sulfonamide
1-[4-(5-methylpyridin-2-yl)-1-phenylbut-3-yn-2-yl]piperidin-4-ol
6-{[4-(2-methylphenyl)phenyl]methyl}-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
(4aS,8aR)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-({8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)benzamide
N-(1H-imidazol-2-ylmethyl)-2-(N-phenylmethanesulfonamido)propanamide
6-[(1R,5S)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
2-benzyl-9-(4,4,4-trifluorobutanoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
4-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyridine
dimethyl({4-methyl-5-[1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
6-(1-benzyl-1H-pyrazol-4-yl)pyridin-3-amine
1-[2-(2,2-diphenylethyl)morpholin-4-yl]-3-(1H-pyrazol-1-yl)propan-1-one
1-cyclohexyl-N-[1-(4-fluorophenyl)-2-hydroxyethyl]piperidine-4-carboxamide
2-[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-methoxyethan-1-one
4-(3-{[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]oxy}benzoyl)morpholine
3-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-4,5,6,7-tetrahydro-1H-indazole
2-cyclopropyl-N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}pyrimidine-5-carboxamide
N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}propanamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-1-[(3R)-3-hydroxypyrrolidin-1-yl]ethan-1-one
N-(furan-2-ylmethyl)-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
2-[benzyl(methyl)amino]-N-[2-(1,3-thiazol-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide