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1-ethyl-3-methyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-1H-pyrazole-4-carboxamide
7-[(3-methylphenyl)methyl]-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
5-{[({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-3-(1H-pyrazol-4-yl)benzamide
5-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
ethyl 1-[5-(3-fluorophenyl)-1,2,4-triazin-3-yl]piperidine-3-carboxylate
1-{1'-[(4-chlorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
1-({1-[6-(3-acetylphenyl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
N-[3-(furan-2-yl)-3-phenylpropyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-3-ol
methyl 6-[(3-methylphenyl)methyl]-2-[(oxolan-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl 3-(1,3-dimethyl-1H-pyrazole-5-amido)-6-{[methyl(thiophen-3-ylmethyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
(3R,4R)-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
2-chloro-3-{[(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amino]methyl}-9-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
2-[1-methyl-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-2-yl]ethan-1-ol
N-(cyclopropylmethyl)-N-(2-methoxyethyl)-6-methylimidazo[1,2-a]pyridine-2-carboxamide
N,3,5,7-tetramethyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-indole-2-carboxamide
4-({2-[2-(4-ethylpiperazin-1-yl)ethoxy]phenyl}methyl)-3-methylpiperazin-2-one
4-(2,4-dioxoimidazolidin-1-yl)-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)benzamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[methyl(prop-2-en-1-yl)amino]methyl}piperidin-2-one
5-[3-(3-methoxypropyl)piperidine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
2-(1-ethylpiperidin-4-yl)-N-methyl-N-(oxan-2-ylmethyl)acetamide
1-(3-fluoro-4-methoxybenzoyl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine
4-[3-(4-cyclopropanecarbonyl-1,4-diazepane-1-carbonyl)phenyl]-2-methylbutan-2-ol
N,5,6-trimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
(1S,5R)-3-(2-aminopyridine-4-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(dimethylamino)-N,4-dimethyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]pyrimidine-5-carboxamide
2-[3-(1H-imidazol-1-yl)propyl]-9-[(5-propylfuran-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-1-[2-(2H-indazol-2-yl)acetyl]piperazine-2-carboxamide
3-[(8-fluoroquinolin-2-yl)formamido]-3-(furan-2-yl)propanoic acid
8-fluoro-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]quinoline-2-carboxamide
1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-4-(thiophen-2-yl)butan-1-one
1-{3-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-oxopropyl}pyrrolidin-2-one
3-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]pyridin-2-ol
3-methanesulfonyl-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
7-(4-cyclopentyl-3-oxopiperazine-1-carbonyl)-1,2,3,4-tetrahydroquinoxalin-2-one
3-{1-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}benzoic acid
8-(oxane-4-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
2-{2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(methylsulfanyl)-6-oxo-1,6-dihydropyrimidine-5-carboxamide
(2-{2-[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
2-methyl-6-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-2,3-dihydropyridazin-3-one
2-benzyl-4-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1,3-thiazole
N-[(3S,4R)-1-(3-aminothiophene-2-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
8-cyclopropanecarbonyl-2-(5-methyl-1,3-oxazole-4-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(2-ethoxyethyl)-N-[2-(3-methylpyridin-2-yl)ethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-methoxy-2,3-dihydro-1H-indene-5-carboxamide
N-(2-oxoazepan-3-yl)-2-(1-propylpiperidin-4-yl)acetamide
2-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
(2R,3R)-3-({[4-(hydroxymethyl)oxan-4-yl]methyl}amino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol