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4-(4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-1-yl)pyrimidin-2-amine
1-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(methylsulfanyl)propan-1-one
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-[(4-phenyloxan-4-yl)methyl]-1,4-dihydropyridine-3-carboxamide
1-{4-[2-(1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-(4-methylphenyl)-5-(pyridin-4-yl)pyrimidin-2-amine
8-(2H-1,3-benzodioxol-5-ylmethyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(2,6-dimethylphenyl)methyl]pyrrolidin-3-yl]methanol
2-methyl-5-{1H-pyrrolo[2,3-b]pyridin-6-yl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
N,2-dimethyl-N-[(3-methylpyridin-2-yl)methyl]-6-(propan-2-yl)pyrimidin-4-amine
N-(2-methylpropyl)-1-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
3-{[cyclopropyl(thiophen-3-ylmethyl)amino]methyl}-7-methyl-1,2-dihydroquinolin-2-one
N-[(5-methylpyrazin-2-yl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
6-(aminomethyl)-N,2-dimethyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrimidin-4-amine
(1H-imidazol-2-ylmethyl)[2-methoxy-1-(pyridin-2-yl)ethyl]methylamine
4-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-2-(2-methoxyethyl)morpholine
3-{3-[5-(1-methoxypropan-2-yl)-3-(piperidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-1-yl]propyl}pyridine
3-(4-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}phenyl)prop-2-yn-1-ol
1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-(1H-pyrazol-1-yl)butan-1-one
5-fluoro-2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridine
(1S,5R)-3-cyclobutanecarbonyl-6-[2-(pyrrolidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
N-(1-benzyl-5-oxopyrrolidin-3-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-(pyridin-3-yl)propanamide
ethyl 4-[(2-chlorophenyl)methyl]-1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidine-4-carboxylate
2-acetamido-N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}acetamide
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyrrolidine-1-sulfonamide
N-[2-(1H-indol-1-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
4-(3-{1-[(4-methoxypyridin-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-3-methylpyridine
N,N-bis(2-hydroxyethyl)-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
2-amino-3-ethyl-N-[(3-phenylphenyl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-(2-{2,7-diazaspiro[4.5]decan-7-yl}-2-oxoethyl)morpholine-3,5-dione
(1-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)methanol
N,5-dipropyl-N-(thiophen-3-ylmethyl)-1,2-oxazole-3-carboxamide
(5S,9aS,9bS)-2-(1-methylpiperidin-4-yl)-5-[4-(methylsulfanyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide
9-(cyclopropylmethyl)-1-methyl-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-benzyl-4-[4-(methylsulfanyl)benzoyl]-1,4-diazepan-6-ol
2-{[1-(3-methylphenyl)-1H-1,3-benzodiazol-2-yl]methoxy}acetic acid
1-(3-chlorothiophene-2-carbonyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(4-chlorophenoxy)pyridine-3-carboxamide
2-(1-ethylpiperidin-4-yl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methyl-1,2-oxazole-4-carboxamide
{3-[(2,4-difluorophenyl)methyl]-1-(3-fluoropyridin-2-yl)piperidin-3-yl}methanol
5-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-2-methoxypyridine
6-(2-chlorophenyl)-N-methyl-N-(pyridin-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[methyl(2-phenylethyl)amino]-N-[(6-methylpyridin-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
(3S,4S)-1-(1-aminocyclopropanecarbonyl)-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
N-[(2,5-dimethylphenyl)methyl]-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
2-(2-methoxyphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide