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(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-(3-hydroxyazetidine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-{[7-fluoro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-4-methylbenzamide
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
3-({4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)phenol
1-{1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-4-yl}piperidin-3-ol
1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidine-4-carbonitrile
2-({3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
3-[3-(piperidine-1-carbonyl)pyridin-2-yl]benzonitrile
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
2-{[(1R)-2-hydroxy-1-phenylethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
ethyl 4-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)piperidine-1-carboxylate
1-[(3aS,6aS)-5-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydropyrrolo[2,3-c]pyrrol-1-yl]-3-methylbutan-1-one
3-{2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
6-(2,4-dimethoxyphenyl)-N,N-dimethylpyridine-2-carboxamide
2-{1-butyl-5-[3-(trifluoromethyl)-1H-pyrazol-5-yl]-1H-1,2,4-triazol-3-yl}acetamide
N-[(5-chlorofuran-2-yl)methyl]-N-(pyridin-4-ylmethyl)cyclopropanamine
2-[5-(1-methylpyrrolidin-2-yl)thiophene-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-({3-methyl-7-[3-(trifluoromethyl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-carboxamide
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}acetamide
N-cyclopropyl-1-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
N-(2,2-dimethyloxan-4-yl)-N-ethyl-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
(4-{[2-(ethylamino)pyrimidin-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
3-({3-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]piperidin-1-yl}methyl)pyridine
N-cyclopropyl-5-[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-{[7-chloro-2-(2,5-dimethoxyphenyl)quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]oxolane-2-carboxamide
methyl N-{[(2S,4S)-4-fluoro-1-[4-(5-methylfuran-2-yl)benzoyl]pyrrolidin-2-yl]methyl}carbamate
N-[(4-ethylphenyl)methyl]-N-methyl-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-cyclopropyl-3-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]propanamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrrole-2-carbonyl)piperidine
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(2-methylpyrimidin-4-yl)-1H-pyrazol-1-yl]acetamide
N-(2-fluorophenyl)-2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
8-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(3-methoxyphenoxymethyl)-N-[(2R)-pyrrolidin-2-ylmethyl]-1H-pyrazole-3-carboxamide
1-{2-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]-4-methylpyrimidin-5-yl}ethan-1-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-2-methylpyrimidine-5-carboxamide
(3aR,6aR)-2-cyclopentyl-N-[2-(2-oxopiperidin-1-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(1S,6R)-9-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-3,9-diazabicyclo[4.2.1]nonan-4-one
8-(2-propoxyphenyl)-2-(pyrrolidin-1-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
ethyl 5-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(1R,2R,4R)-N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methylbicyclo[2.2.1]hept-5-ene-2-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}acetamide
1-{2-[1-(1-benzofuran-2-ylmethyl)piperidin-2-yl]ethyl}-4-methylpiperazine
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-[2-(quinolin-8-yloxy)ethyl]acetamide
(1R)-1-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]butane-1,4-diamine
1-(2,1,3-benzoxadiazol-5-ylmethyl)-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
1-methyl-8-(morpholine-4-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[(1,4-dimethyl-1H-pyrazol-5-yl)methyl]-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
N-[(3R,4S)-4-(propan-2-yl)-1-(4-sulfamoylbenzoyl)pyrrolidin-3-yl]acetamide