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4-[2-(dimethylamino)-2-(3-fluorophenyl)acetamido]-N-ethylpiperidine-1-carboxamide
4-[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-5-methyl-1,3-oxazole
1-[3-(1H-pyrazol-5-yl)phenyl]-3-[1-(thiophen-2-ylmethyl)piperidin-4-yl]urea
N-ethyl-2-[4-(2-phenoxyethyl)piperazin-1-yl]pyridine-4-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(phenylamino)pyrimidine-5-carboxamide
6-methyl-N4-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]pyrimidine-2,4-diamine
(3S,4S)-1-[3-(dimethylamino)benzoyl]-4-methylpiperidine-3,4-diol
methyl 1-benzyl-5-{[(5-methylfuran-2-yl)methyl]amino}-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-[(6-methylquinolin-5-yl)methyl]pyrrolidin-3-yl]methanol
(2S,4R)-N,N-diethyl-4-(4-{[methyl(pyrrolidine-1-carbonyl)amino]methyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
[(3S,5R)-5-[(dimethylamino)methyl]-1-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-3-yl]methanol
1-[2-(2-methoxyethyl)morpholin-4-yl]-2-(2,3,6-trimethylphenoxy)ethan-1-one
5-[3-(4-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-1-phenyl-1H-1,2,3,4-tetrazole
N4-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
5-ethyl-N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-1,3,4-oxadiazol-2-amine
1-cycloheptyl-6-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
2-(5-{[2-(ethylsulfanyl)-1,3-thiazol-4-yl]methyl}-3-methyl-1H-1,2,4-triazol-1-yl)pyridine
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]pyrimidine-5-carboxamide
6-methoxy-2-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-1,2,3,4-tetrahydroisoquinoline
1-(cyclopropylmethyl)-3-(2-methylquinolin-5-yl)-6-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-ethyl-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
methyl 5-[2-(1H-imidazol-2-yl)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
ethyl 3-[(3-chlorophenyl)methyl]-1-[3-(1H-imidazol-2-yl)benzoyl]piperidine-3-carboxylate
1-{2-[benzyl(methyl)amino]acetyl}-1,4-diazepane-6-carboxylic acid
N-cyclopropyl-2-[2-(3-methylbut-2-en-1-yl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]pyridine-4-carboxamide
5-[4-oxo-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridine-2-carbonitrile
N,N-dimethyl-3-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]aniline
3-[({2-[4-(dimethylamino)phenyl]ethyl}amino)methyl]piperidin-3-ol
5-[2-(3-fluorophenyl)-3-oxopiperazine-1-carbonyl]thiophene-2-carboxylic acid
5-[4-(diphenylmethyl)piperazine-1-carbonyl]-2-methylpyrimidine
4-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
benzyl (7S,9aR)-6,9-dioxo-7-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-[4-(3-methoxyphenyl)phenyl]-1-propylpiperidine-3-carboxamide
6-(2,3-dihydro-1-benzofuran-2-carbonyl)-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
(2S,4R)-4-(4-{[1-(3-chloro-2-fluorophenyl)-N-methylformamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
2-(4-fluorophenyl)-2-hydroxy-N-[(1r,4r)-4-methoxycyclohexyl]acetamide
4-(2,5-dimethoxybenzoyl)-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
2-[8-(3-methoxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-1,3-thiazole-4-carboxamide
methyl 5-(cyclobutylamino)-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[2-(3-methyl-4-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}-1H-pyrazol-1-yl)ethyl]thiomorpholine
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4-methylpiperazine
N-methyl-5-({[2-(methylsulfanyl)ethyl]amino}methyl)-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
4-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
1-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-[(8-methoxy-2H-chromen-3-yl)methyl]-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
methyl 3-(2-chlorobenzenesulfonamido)-5-[(cyclopropylformamido)methyl]benzoate