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(3R,9aR)-3-benzyl-8-[(3-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(1R,2S)-2-phenylcyclopropyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
4-[(4-fluorophenyl)methyl]-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
6-(2-chlorophenyl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[2-(morpholin-4-yl)ethyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
3-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1H-pyrazol-1-yl)propanoic acid
2-ethoxy-4-{[methyl({2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})amino]methyl}phenol
4-[3-(2-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-phenylpiperidine-4-carbonitrile
(5-{[4-(5-chloropyridin-2-yl)piperazin-1-yl]methyl}-2-ethoxyphenyl)methanol
dimethyl(2-{2-[1-(quinolin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-{3-[benzyl(methyl)amino]piperidin-1-yl}-6-methylpyridine-3-carbonitrile
(3R,4R)-4-(morpholin-4-yl)-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-3-ol
(2-methoxyethyl)[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl][(1-methyl-1H-pyrazol-4-yl)methyl]amine
2-[2-({3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]pyrimidine
2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-(furan-2-ylmethyl)-N-methylacetamide
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
1-(4-{[3-(2-methylphenoxy)azetidin-1-yl]methyl}phenyl)ethan-1-one
1-ethenyl-N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methyl-1H-pyrazole-4-carboxamide
4-{4-[(4-fluorophenyl)methyl]-6-hydroxy-1,4-diazepan-1-yl}-4-oxobutanoic acid
4-[(1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-2-yl)methyl]morpholine
4-{[4-(benzyloxy)phenyl]methyl}morpholine-2-carboxamide
2-[1-(dimethyl-1,3-thiazol-2-yl)-1H-pyrazol-4-yl]-6-fluoro-N,N-dimethylquinoline-4-carboxamide
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]pyridine
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2-(dimethylamino)-2-(2-fluorophenyl)-N-methylacetamide
methyl 5-[(3S,4R)-3-acetamido-4-(4-methylphenyl)pyrrolidin-1-yl]-5-oxopentanoate
4-({4-methyl-5-[1-(pyridine-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-cyclopropyl-4-phenyl-9-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-propyl-N-(pyridin-3-ylmethyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-pyrazole-5-carboxamide
N-[2-(3-methoxyphenyl)phenyl]-1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-[ethyl(methyl)amino]propanamide
N-benzyl-N-ethyl-3-{[(3S)-2-oxoazepan-3-yl]amino}propanamide
N-[(2,4-dichlorophenyl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
2-[4-(2-methoxybenzoyl)piperazin-1-yl]-4-(3,3,3-trifluoropropyl)pyrimidine
1-(6-aminopyrimidin-4-yl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
2-{3-[(2-butylpyrrolidin-1-yl)methyl]phenoxy}ethan-1-ol
N-[(2-methoxyphenyl)methyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(cyclohex-1-ene-1-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
ethyl (4aR,6R,8aS)-6-(morpholin-4-yl)-2-(1H-pyrrole-2-carbonyl)-decahydroisoquinoline-8a-carboxylate
2-(dimethylamino)-4-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}pyrimidine-5-carboxamide
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidine
3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-N-(1-methyl-1H-indazol-3-yl)benzamide
2-(pyridin-3-yl)-4-(1,3-thiazol-4-ylmethyl)morpholine
5-(oxolan-2-yl)-3-{[4-phenyl-5-(thiophen-3-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
N-cyclopropyl-1-{1-[(4-methoxypyridin-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-methyl-1,3-thiazole-5-carboxamide
5-methoxy-3-methyl-2-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}-1H-indole
5-ethyl-2-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)pyrimidin-4-amine
N-[(2-fluorophenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine