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5-{4-[(4-ethyl-3-oxopiperazin-1-yl)methyl]phenoxymethyl}furan-2-carboxylic acid
4-{[4-(trifluoromethyl)phenyl]methyl}-1,4-oxazepan-5-one
1-[2-(benzenesulfonyl)ethyl]-1,2-dihydroquinoxalin-2-one
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
7-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1,3-diazepane-2,4-dione
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-4-yl)propanamide
2-{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}-1,2-oxazolidine
1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-3-(1H-pyrazol-4-yl)propan-1-one
6-tert-butyl-1-methyl-N-[2-(oxan-3-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3aS,7aR)-2-(2-{[(3,5-dimethylphenyl)methyl]sulfanyl}acetyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
[(1-ethyl-1H-pyrazol-4-yl)methyl][(1-ethylpyrrolidin-2-yl)methyl]{[1-(2-methoxyethyl)piperidin-4-yl]methyl}amine
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-3-(1H-pyrazol-1-yl)benzamide
7-(2,2-dimethylpropyl)-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-N-methylbenzene-1-sulfonamide
4-chloro-2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-methyl-1H-indole
({4-[1-(dimethylamino)ethyl]phenyl}methyl)[2-(1H-imidazol-1-yl)ethyl]methylamine
3-(2,3-dihydro-1H-isoindole-2-carbonyl)-4-fluorobenzene-1-sulfonamide
3-chloro-4-fluoro-N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-1-benzothiophene-2-carboxamide
(3S,4R)-1-(5-acetyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-6-({4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-(4-oxo-4-phenylbutanoyl)piperidine-4-carboxylate
3-(1-{[4-(propan-2-yloxy)phenyl]methyl}piperidin-3-yl)-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-{3-[2-methyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]-3-oxopropyl}acetamide
9-methoxy-N-[(2-methoxyphenyl)methyl]-3-[(3-methylthiophen-2-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(3-fluoro-4-methoxybenzenesulfonyl)-4-(hydroxymethyl)azepan-4-ol
2-{4-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1H-pyrazol-1-yl}-N-(1-methyl-1H-pyrazol-5-yl)acetamide
(1S,3R)-N-(cyclohex-1-en-1-ylmethyl)-3-[3-(thiophen-3-yl)propanamido]cyclopentane-1-carboxamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-2-oxo-2-phenylacetamide
2-(dimethylamino)-N-[2-(4-hydroxyphenyl)ethyl]-2-(2-methylphenyl)acetamide
2-amino-4-(3-chloro-4,5-diethoxyphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(4-chloro-1H-pyrazole-3-carbonyl)-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
1-[(3,5-difluorophenyl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
(3aS,6aS)-2-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-methyl-5-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
2-[2-(butan-2-yl)phenoxy]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)acetamide
N-[3-(azepan-1-yl)propyl]-N-methyl-[1,2,4]triazolo[4,3-a]pyridine-7-carboxamide
6-amino-1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]hexan-1-one
2-{2-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-6-methylpyridine
4-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}phenol
2-(2-methoxyethyl)-8-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3-{1-[1-(benzenesulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-1-ol
(4aS,7aR)-1-{2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]acetyl}-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}piperidin-1-yl)acetamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
9-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(2-methoxyethyl)-4-[(3-phenoxyphenyl)methyl]morpholine
N-(oxan-4-ylmethyl)-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4-(2-phenoxyethyl)piperidin-4-yl)methanol
1-[3-(methylsulfanyl)propyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide