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N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2,2-dimethyloxane-4-carboxamide
N-(furan-2-ylmethyl)-N,1-dimethyl-5-[(3-methylbutyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(pyridin-4-yl)ethyl]piperidine-3-carboxamide
4-(3-chlorophenyl)-3-(4-hydroxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 3-[(4-fluorophenyl)methyl]-1-(2-methylpropanoyl)piperidine-3-carboxylate
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-(1,3,4-thiadiazol-2-yl)urea
3-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-methyl-1H-indole
9-methoxy-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{3-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]phenoxy}acetamide
6-methoxy-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,3-dihydro-1H-indene-5-carboxamide
2,5-dimethyl-N-({7-[(2,3,6-trifluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)furan-3-carboxamide
4'-(pyrrolidin-3-ylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-amine
1-[(2-chlorophenyl)methyl]-4-[(1s,4s)-4-aminocyclohexyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[3-(azepan-1-yl)-2-hydroxypropyl]quinoxaline-5-carboxamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
5-ethoxy-2-methyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1-benzofuran-3-carboxamide
2-[5-(3-chloro-2,4-difluorophenyl)-4-phenyl-1H-imidazol-1-yl]-N-methylacetamide
methyl 4-(4-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(2,5-difluorophenyl)methyl]-5-methoxybenzamide
5-chloro-2-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
2-{[5-(1,5-dimethyl-1H-pyrazol-3-yl)-4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
4-(2-methoxypyridin-3-yl)pyridin-2-amine
{5-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
8-methoxy-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[4-(3-methoxybenzoyl)piperazin-1-yl]propan-1-one
2-methoxy-N-(1-{1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
5,5-dimethyl-1-{2-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
7-cyclohexyl-2-[2-(pyridin-2-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-1-[(2-methoxynaphthalen-1-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-(naphthalen-1-yl)-5-{1-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-imidazol-2-yl}pyrimidine
dimethyl({4-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,3-thiazol-2-yl}methyl)amine
5-methanesulfonyl-2-[(4-methoxyphenyl)methyl]-4-(piperidin-3-yl)pyrimidine
9-(2-methoxyquinoline-4-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
6-(furan-3-carbonyl)-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-cyclohexyl-3-methyl-N-(pyridin-3-ylmethyl)-1,2-oxazole-5-carboxamide
1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-methyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
[(1-ethyl-1H-pyrazol-4-yl)methyl][(1-methyl-1H-imidazol-2-yl)methyl](2-methylpropyl)amine
1-methyl-3-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
2-(adamantan-1-yl)-4-hydroxy-N-methyl-N-(1-methylpiperidin-4-yl)pyrimidine-5-carboxamide
[4-(2-amino-4-methyl-1,3-benzothiazol-6-yl)phenyl]methanol
7-(2,6-dimethoxyphenyl)-9-methoxy-4-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3E)-N-[(4-methoxyphenyl)methyl]-N-propylhex-3-enamide
2-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
2-cyclopropyl-N-[(4-methoxyphenyl)methyl]-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
ethyl 3-(2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamido)propanoate
3-cyclohexyl-N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1H-pyrazole-4-carboxamide
5-[4-(2-ethoxyethyl)piperazine-1-carbonyl]-2-(pyridin-2-yl)pyrimidin-4-ol
N-(1-methyl-1H-1,3-benzodiazol-2-yl)-5-[1-(propan-2-yl)pyrrolidin-2-yl]thiophene-2-carboxamide