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5-[1-(4-methylbenzoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
2-amino-8-(3-chloro-5-fluoro-4-methoxyphenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
6-[(oxan-3-yl)amino]-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
N-cyclopropyl-2-ethyl-N-({3-[(1-methylpiperidin-3-yl)methoxy]phenyl}methyl)butanamide
1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
1-[2-(3-fluorophenyl)ethyl]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-6-oxopiperidine-3-carboxamide
3-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-1-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}urea
2-(2-hydroxyethyl)-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
6-{5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-phenyl-1H-imidazol-1-yl}-2-methylheptan-2-ol
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-3-methoxypropan-1-one
5-methyl-N-[3-(pyridin-4-yl)propyl]-4-{[1-(thiophen-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
3-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-N-(pyridin-3-yl)benzamide
2-{[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]methyl}quinolin-4-ol
(2-methylpropyl)(pyridin-2-ylmethyl){[4-(pyrimidin-5-yl)phenyl]methyl}amine
N,1,3-trimethyl-2,6-dioxo-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
6-[(4aS,8aR)-1-(4-hydroxybutyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]pyridine-2-carbonitrile
2-[methyl({[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl})amino]-1-phenylethan-1-ol
3-[3-({[1-(3,4-dimethylphenyl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(pyrrolidin-1-yl)propan-1-one
4-[({1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}carbamoyl)amino]-N-propylbenzamide
5-[4-(4-chlorophenyl)butanoyl]-1-methyl-N-[3-(morpholin-4-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(4-fluorophenyl)methyl]-4-(2-methylpyrimidin-4-yl)-2-(propan-2-yl)-1,4-diazepane
1-{2-[2-(3-fluorophenyl)piperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1-(pyrimidin-2-yl)piperidin-3-amine
8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[(3R,4S)-1-[(2-aminopyridin-3-yl)methyl]-4-propylpyrrolidin-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
4-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
5-{[(2-methylpropyl)carbamoyl]carbonyl}-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-methyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1H-indole-6-carboxamide
2-fluoro-N-{2-[1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]ethyl}benzamide
3-cyclobutyl-5-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[(3-fluorophenyl)methyl]-6-oxo-N-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-3-carboxamide
(5-{1-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)methanol
1-{3-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]piperidin-1-yl}propan-1-one
1-(3-methoxyphenyl)-4-[3-(4-methoxyphenyl)propanoyl]piperazin-2-one
3-(2-amino-1,3-thiazol-4-yl)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]propanamide
7-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(pyridine-4-carbonyl)-1,4-diazepane
N,1,4,6-tetramethyl-2-oxo-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-1,2-dihydropyridine-3-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
2-fluoro-N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-5-sulfamoylbenzamide
1-cyclohexyl-4-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
8-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[3-hydroxy-1-(2-methoxyethyl)-2-oxopiperidin-3-yl]methyl}-1λ6-thiomorpholine-1,1-dione
4-[3-(cyclopropylmethyl)-5-(1H-imidazol-1-ylmethyl)-1H-1,2,4-triazol-1-yl]-3-methylpyridine
4-{1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl}-2-(pyridin-4-yl)pyridine
1-methyl-N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]-1H-imidazole-5-carboxamide