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N-(4-chloro-3-methylphenyl)-2-({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amino)acetamide
3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide
6-methoxy-N,3-dimethyl-N-[3-(3-methylphenoxy)propyl]-1-benzofuran-2-carboxamide
2-(2,3-difluorophenoxymethyl)-N-[(3-methoxyphenyl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-3-(3-methoxypropyl)piperidine-3-carboxylic acid
2-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-4,5,6,7-tetrahydro-1,3-benzothiazole
6-{4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}quinoxaline
methyl 2-[1-(2-methoxyethyl)-2,4-dioxo-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
1-{[3-(azepane-1-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-3-ol
[(3R,5R)-5-(morpholin-4-ylmethyl)-1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]methanol
N-(2-ethyl-3-methyl-1-benzofuran-7-yl)-4-methanesulfonylpiperazine-1-carboxamide
(2S)-2-amino-1-[6-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]butan-1-one
4-chloro-2-({3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(2-methylphenyl)piperidine
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-N'-(3-methylphenyl)propanediamide
1-[3-(2-methylphenoxy)azetidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-[2-methyl-5-(3-methylbutanamido)phenyl]-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
1-(4-{[4-(4-fluorophenoxy)piperidin-1-yl]methyl}phenyl)ethan-1-one
1-(azocan-1-yl)-3-(5-methoxy-2-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}phenoxy)propan-2-ol
2-methyl-N-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)oxane-2-carboxamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[2-(2,4-dimethoxyphenyl)ethyl]acetamide
2-{4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
1-ethyl-N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-1H-pyrazole-3-carboxamide
6-{[3-(pyridin-2-yl)azetidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroquinolin-2-one
9-ethyl-4-[3-(4-fluorophenoxy)propyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(2-hydroxy-1-phenylethyl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-{3-[(2,6-dichlorophenyl)methyl]-5-(morpholin-3-ylmethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
(4aR,7aS)-1-[(2-ethoxyphenyl)methyl]-4-(1H-imidazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({3-methyl-7-[2-(1H-pyrazol-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-3-yl)acetamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
3-(4-fluorophenyl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
[(3R,4R)-1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
propan-2-yl 4-chloro-3-({[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]carbamoyl}amino)benzoate
4-ethyl-3-[1-(2-methyl-1,8-naphthyridine-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[4-(6-methylpyridin-3-yl)benzenesulfonyl]thiomorpholine
3-(3-cyano-4-methylphenyl)-1-(oxan-4-yl)urea
4-(1-ethylpiperidin-3-yl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
2-methoxy-1-{9-[3-(morpholin-4-yl)azetidin-1-yl]-3-azaspiro[5.5]undecan-3-yl}ethan-1-one
N-({7-[2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-2-yl)acetamide
5-(2-chloro-4-fluorophenoxymethyl)-N-(3-phenylpropyl)-1,2-oxazole-3-carboxamide
8-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[3-(5-benzyl-4-phenyl-1H-imidazol-1-yl)propyl]pyrrolidin-2-one
1-methanesulfonyl-3-[4-(trifluoromethyl)benzoyl]piperidine
(1S,5R)-6-(cyclobutylmethyl)-3-(4-fluoro-3-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
5-{3-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-4-methylpyrimidine
2-[(3-methoxyphenyl)methyl]-N,N-dimethyl-3-oxo-2,8-diazaspiro[4.5]decane-8-sulfonamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1H-1,2,4-triazole-5-carboxamide