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4-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyridin-2-amine
4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-amine
2-{6-chloro-[1,2,4]triazolo[4,3-a]pyridin-3-yl}-6-methylpyridine
(1R,9aR)-1-[4-(2-methoxyethyl)phenoxymethyl]-octahydro-1H-quinolizine
2-methoxy-N-({5-[(2,3,4-trifluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
1-[3-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-oxopropyl]azepan-2-one
ethyl 1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-(2-phenylethyl)piperidine-4-carboxylate
2-chloro-4-{[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]methyl}phenol
3-fluoro-4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)pyridine-3-carboxamide
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-(3-methoxyphenoxymethyl)piperidine
3-chloro-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
N-[(2-aminopyrimidin-5-yl)methyl]-N-methyl-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
5-methyl-1-(2-methylphenyl)-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazin-2-one
8-(8-hydroxyquinoline-7-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-1H-1,2,3-triazole-5-carboxamide
4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidine
N-ethyl-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
1-(3-methoxypropyl)-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
ethyl 4-{[(4-oxo-4H-chromen-6-yl)carbamoyl]amino}piperidine-1-carboxylate
ethyl 5-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
methyl({[2-(propylsulfanyl)pyrimidin-5-yl]methyl}){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
(4aS,8aR)-1-(2-aminoethyl)-6-[3-(pyridin-3-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
1-{5-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
2-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-5,6-dimethylpyridine-3-carbonitrile
(2S)-2-amino-1-{7-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}butan-1-one
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-1-[2-(pyridin-3-yl)piperidin-1-yl]propan-1-one
(3S,4S)-3-hydroxy-4-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-1H-imidazol-1-yl]-1λ6-thiolane-1,1-dione
1-(1-methylpiperidin-4-yl)-3-phenyl-1-(2-phenylethyl)urea
1-methyl-N-(oxolan-2-ylmethyl)-3-propyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-5-carboxamide
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(3S)-2-oxoazepan-3-yl]benzamide
3-chloro-6-(4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)pyridazine
(4aS,7aR)-1-cyclopropanecarbonyl-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
[1-(2-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)piperidin-3-yl]methanol
6-fluoro-2-{[(2S)-2-(piperidine-1-carbonyl)pyrrolidin-1-yl]methyl}quinolin-4-ol
(1R,5R)-3-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-({[(1S,2S)-1,3-dihydroxy-1-phenylpropan-2-yl]carbamoyl}amino)-N,N,2-trimethylbenzamide
2-cyclopropyl-N-(pyridin-3-ylmethyl)-1,3-benzoxazole-6-carboxamide
N-(3-fluorophenyl)-6-[2-(4-phenylphenyl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
3-methyl-1-propyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H-pyrazole-4-carboxamide
ethyl 1-(benzylcarbamoyl)-4-(2-phenylethyl)piperidine-4-carboxylate
4-[2,5-dimethoxy-4-(methylsulfanyl)phenyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4,6-dimethyl-N-{[2-(trifluoromethoxy)phenyl]methyl}pyrimidin-2-amine
N-[2-(dimethylamino)ethyl]-3-{1-[(3-ethoxyphenyl)methyl]piperidin-4-yl}propanamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetamide
N-cyclopropyl-N-{[4-(methylsulfanyl)phenyl]methyl}-2-(propan-2-yloxy)propanamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
N-[2-(4-chlorobenzenesulfonamido)ethyl]-2-(methylamino)pyridine-3-carboxamide
1-ethyl-8-[1-(methylsulfanyl)propan-2-yl]-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione