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(2R,6S)-4-{1-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}-2,6-dimethylmorpholine
1-(propan-2-yl)-3-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}piperidine
9-(5-chloropyridin-2-yl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-5-phenylpentane-1,5-dione
1-{6-[4-(3-methylphenoxy)piperidin-1-yl]pyridin-2-yl}ethan-1-ol
N-butyl-3-(3,4-dimethoxyphenyl)-N-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
3-benzyl-1-methyl-3-[3-oxo-3-(piperidin-1-yl)propyl]-2,3-dihydro-1H-indol-2-one
4-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-methyl-2-phenyl-2-({[1-(propan-2-yl)-1H-pyrazol-4-yl]carbamoyl}amino)acetamide
3-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
5-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}-2-(2-methoxyethyl)pyrimidine
2-(pyridin-3-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]pyrimidine-5-carboxamide
(2R,3R,6R)-5-(1H-1,2,3-benzotriazole-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
6-(2-methoxyphenyl)-1,3-benzothiazol-2-amine
5-(2-chloro-4-methoxyphenoxymethyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,2-oxazole-3-carboxamide
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2,6-dimethylpyrimidine-4-carboxamide
6-methyl-2-[1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
benzyl({[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})[(4-methyl-1,3-thiazol-5-yl)methyl]amine
1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-4-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,4-dihydropyridine-3-carboxamide
6-[3-(4-chloro-2-methylbenzoyl)piperidine-1-carbonyl]quinoline
1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-ol
(3S,4S)-1-(1,4-dimethylpiperidine-4-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
6-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-2-(2-methoxyethyl)-1,3-benzoxazole
5-methyl-1-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-5-phenylpiperidin-2-one
9-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(2,6-dimethylphenoxymethyl)-N-[(1R,2S)-2-phenylcyclopropyl]-1,2-oxazole-3-carboxamide
4-(1H-imidazol-1-yl)-1-[2-(3-methoxypropyl)piperidin-1-yl]butan-1-one
5-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3,5,7-trimethyl-2-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1H-indole
2-(2-methoxyethyl)-9-(2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
7-methyl-6-(3-methyl-1H-pyrazole-5-carbonyl)-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
2-methyl-3-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-2,8-diazaspiro[4.5]decane
N-(3-methoxy-2,2-dimethylpropyl)-2,2,3,3-tetramethylcyclopropane-1-carboxamide
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N3-(4-fluorophenyl)-N5-[(4-methylphenyl)methyl]piperidine-3,5-dicarboxamide
4-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-[3-(trifluoromethyl)phenyl]pyrimidine
3,4-dimethoxy-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)benzamide
6-cyclopropyl-2-(3-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
2-{[benzyl(ethyl)amino]methyl}pyridine-3-carboxylic acid
3-(4-ethyl-1H-pyrazol-5-yl)-1-(naphthalen-1-ylmethyl)piperidine
1'-(1H-pyrazole-4-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]
1-(3-{[2-(methoxymethyl)piperidin-1-yl]sulfonyl}benzoyl)piperazine
3-chloro-N-cyclopentyl-4-{[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]oxy}benzamide
7-acetamido-1-[2-(pyridin-2-yl)ethyl]-N-[2-(thiophen-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
5-[(2E)-but-2-en-1-yl]-N-[(4-methoxyphenyl)methyl]-N-methyl-1,3,4-oxadiazole-2-carboxamide
4-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidine-1-carbonyl)-1-oxaspiro[4.5]decan-2-one
4-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-1-(3-methoxyphenyl)piperazin-2-one
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}-3-(methylsulfanyl)propanamide
7-fluoro-2-methyl-N-[2-(pyridin-3-yloxy)propyl]quinoline-4-carboxamide