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1-(3-ethyl-1,2-oxazole-5-carbonyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
2-cyclopropyl-9-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 1-(2-methoxyethyl)-5-[(1-methylpiperidin-4-yl)amino]-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1R,5R)-6-(cyclopropylmethyl)-3-{[5-(1H-pyrazol-5-yl)furan-2-yl]sulfonyl}-3,6-diazabicyclo[3.2.2]nonane
6-methyl-4-{2-methyl-2,7-diazaspiro[4.5]decane-7-carbonyl}-1,2-dihydroquinolin-2-one
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-(4-methyl-1,4-diazepan-1-yl)propan-1-one
(3R)-3,4,4-trimethyl-1-(pyrimidin-5-ylmethyl)pyrrolidin-3-ol
1-{2-oxo-2-[2-(2-phenylethyl)piperidin-1-yl]ethyl}piperidine-4-carboxamide
N-tert-butyl-2-{4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-ylmethyl]phenoxy}acetamide
2-({4-benzyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)benzoic acid
1-ethyl-6-oxo-N-(pyridin-3-yl)piperidine-3-carboxamide
2-(propan-2-yl)-9-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 1-ethoxy-2-oxo-8-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
ethyl 5-[2-(1H-imidazol-2-yl)benzoyl]-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(2E)-1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-phenylprop-2-en-1-one
3-(4-{1-[2-(3-methylpyridin-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}phenyl)prop-2-yn-1-ol
(1S,5R)-3-[2-(5-acetylthiophen-3-yl)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-butyl-4-(3-methyl-1H-pyrazole-5-carbonyl)-1-(3-phenylphenyl)piperazin-2-one
5-ethyl-5-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
5-{1-[2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-[(2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}-7-(methylsulfanyl)quinolin-3-yl)methyl]-N-(oxolan-2-ylmethyl)furan-2-carboxamide
1-(1-benzothiophene-2-carbonyl)azepan-4-amine
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-[(2-methylphenyl)sulfanyl]ethan-1-one
(3aR,6aR)-2-(cyclobutylmethyl)-5-(2,4-dimethylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(3R,4S)-1-(2-chloro-5-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
3-{[(3R)-3-hydroxypyrrolidin-1-yl]sulfonyl}-N-[(5-methylpyrazin-2-yl)methyl]benzamide
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamide
5-methoxy-2-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-1-methyl-1H-indole
methyl (2S)-1-({6-[methyl(2-phenylethyl)carbamoyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)pyrrolidine-2-carboxylate
4-(3-benzyl-1H-pyrazol-5-yl)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
2-(1-propylpiperidin-4-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(pyrazin-2-yl)pyrrolidin-3-yl]acetamide
6-ethyl-2-methyl-N-(2-oxopyrrolidin-3-yl)quinoline-4-carboxamide
5-(2,1,3-benzoxadiazol-4-ylmethyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
5-methyl-N-{1-[2-(trifluoromethyl)phenyl]ethyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-2,1-benzoxazole
(1S,2S,9R)-11-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
N-ethyl-2-[4-(4-methylphenyl)piperazin-1-yl]pyridine-3-carboxamide
5-(1-benzyl-1H-pyrazole-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-methyl-5-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-1H-pyrazole
6-cyano-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(furan-3-ylmethyl)pyrrolidin-3-yl]pyridine-3-carboxamide
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-{[1-(6-cyanopyridin-2-yl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
3-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-N-(pyridin-3-yl)propanamide
(3R,4S)-4-cyclopropyl-1-[6-(3-fluorophenyl)pyridine-3-carbonyl]pyrrolidin-3-amine
N-[2-(2-fluorophenyl)ethyl]-5-methyl-4-[4-(morpholin-4-yl)piperidin-1-yl]thieno[2,3-d]pyrimidine-6-carboxamide