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1,9-dimethyl-4-{[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]methyl}-1,4,9-triazaspiro[5.5]undecane
4-[(5-methylfuran-2-yl)methyl]-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
N-cyclopropyl-N-(1-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
3-{[methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}quinolin-7-ol
3-[({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]propanamide
1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
1-[3-(3-methoxyphenoxy)azetidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
1-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propane-1,2-dione
N-[2-(3-methoxy-4-propoxyphenyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]imidazo[1,2-a]pyridine-6-carboxamide
N-benzyl-2-{4-[4-(4-formyl-1,4-diazepan-1-yl)piperidin-1-yl]phenyl}acetamide
3-[(3-chlorophenyl)methyl]-N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
1-(4-methoxyphenyl)-4-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}piperazin-2-one
3-[(3R,4S)-4-(dimethylamino)-1-[(1-methyl-1H-1,2,3-benzotriazol-4-yl)sulfonyl]piperidin-3-yl]propan-1-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-9-methoxy-7-oxo-3-[2-(pyridin-3-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
methyl 2-[(4-chlorophenyl)sulfamoyl]-6-(2-methylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-benzyl-2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)acetamide
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
3-(azocan-1-yl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}propanamide
5-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1-methyl-3-phenyl-1H-pyrazole
3-[(3R,4S)-1-[5-(ethylcarbamoyl)pyridin-2-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N2,N2-dimethyl-N4-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
3-methyl-8-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-3-hydroxy-1,2-oxazole-5-carboxamide
1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(3E)-5,5-dimethyl-2-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}hex-3-enoic acid
3-{4-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}propanamide
1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 6-benzoyl-2-[methyl(2-phenylethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(5-fluoro-1-methyl-1H-indazol-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-({5-carboxy-1-ethyl-1H-pyrrolo[2,3-c]pyridin-3-yl}methyl)-3-propylpiperidine-3-carboxylic acid
4-(cyclohexylmethyl)-1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
6-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
3-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
(2S,4R)-4-{[(4-phenylphenyl)methyl]amino}-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
3-{[2-(2,2-diphenylethyl)morpholin-4-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
2-{4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}pyridin-4-amine
4-{1-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-methylpropan-2-yl}morpholine
N-propyl-7-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[1-(furan-2-ylmethyl)piperidin-4-yl]-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-amine
ethyl 2-(4-carbamoylphenyl)pyridine-3-carboxylate
2-amino-6-methyl-4-(1-phenyl-1H-pyrazol-5-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-[4-(4-methoxyphenyl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
1-(dimethylamino)-2-[4-(2-ethylbutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-2-ol
N-(prop-2-en-1-yl)-3-{[1-(pyridin-4-yl)propyl]sulfamoyl}benzamide
3-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-[2-(piperidin-1-ylmethyl)phenyl]urea
(5S,9aS,9bS)-5-(1H-pyrazol-3-yl)-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-oxo-N-[2-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decane-8-carboxamide
(1S,5R)-3-(7-fluoro-4-methylquinolin-2-yl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one