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N'-[2-(2-fluorophenoxy)ethyl]-N-[2-(methylsulfanyl)phenyl]butanediamide
(3S,4S)-N-(4-chloro-2-fluorophenyl)-3,4-bis(hydroxymethyl)pyrrolidine-1-carboxamide
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
1-[(3,4-dimethylphenyl)methyl]-4-{2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperazin-2-one
2-(furan-2-yl)-1-(2-methyl-1-benzofuran-5-carbonyl)pyrrolidine
8-[4-(1H-indol-3-yl)butan-2-yl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{3-ethyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-N-[2-(4-fluorophenyl)ethyl]acetamide
1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-2-(propan-2-ylsulfanyl)ethan-1-one
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
5-{5-methylimidazo[1,2-a]pyridin-2-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-benzoyl-1-(2,4-difluorobenzoyl)piperidine
(4aR,7aS)-1-(2-methoxyacetyl)-4-[2-(pyridin-3-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1'-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
2-methyl-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1S,5R)-6-benzyl-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
dimethyl[2-(2-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]amine
1-[2-(dimethylamino)ethyl]-3-(3-methoxyphenyl)-3-[2-(3-methoxypiperidin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1λ6-thiomorpholine-1,1-dione
N-(2,3-dimethylphenyl)-3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
4-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]pyridin-2-amine
(1S,5R)-6-(1H-indole-6-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[5-(3-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)thiophen-2-yl]ethan-1-one
1-[2-(4-methoxyphenyl)ethyl]-5-(4-methylpiperazine-1-carbonyl)piperidin-2-one
1-(2-chloropyridin-3-yl)-3-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)urea
1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-phenyl-4-(4-phenylbutanoyl)piperazin-2-one
5-(methoxymethyl)-N-methyl-N-(quinoxalin-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[(5-methylfuran-2-yl)methyl]benzamide
(1S,5R)-3-cyclobutanecarbonyl-N-(2-phenylethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-(pyrazine-2-carbonyl)-1,4-diazepan-6-yl]oxy}acetamide
(3aR,6aR)-2-acetyl-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-(4-{[3-(5-methylfuran-2-yl)phenyl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
1-[4-(2,3-dihydro-1H-isoindole-2-carbonyl)phenyl]imidazolidine-2,4-dione
1-(2-methanesulfonylethyl)-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperazine
3-[(4aR,7aS)-4-(cyclohexylcarbamoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
(1R,7S)-3-tert-butyl-N-methyl-4-oxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[(2R,3R)-1'-(furan-2-ylmethyl)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
(1S,5R)-3-[(4-chloro-2-fluorophenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,4R)-4-(3-methoxyphenyl)-1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidine-3-carboxylic acid
4-{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}morpholine
(3S,4S)-1-(1-benzoylpiperidin-4-yl)-4-(4-fluorophenyl)piperidin-3-ol
ethyl 1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
5-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-1-methyl-1H-imidazole
N-{[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-[(5-methylthiophen-2-yl)methyl]acetamide
3-cyclopropyl-4-(5-fluoro-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3,3-diethyl-1-[(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]-1-{[(2S)-5-oxopyrrolidin-2-yl]methyl}urea