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N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
4-[1-benzyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]-1λ6-thiane-1,1-dione
N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-methyl-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[3-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid
(2H-1,3-benzodioxol-4-ylmethyl)[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)amine
6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purin-2-amine
2-cyclopentyl-N-{[(2S,4S)-4-fluoro-1-[(3E)-pent-3-enoyl]pyrrolidin-2-yl]methyl}acetamide
3-(3,4-difluorophenyl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]propanamide
9-methoxy-N-[(3-methoxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
ethyl 4-{[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]amino}piperidine-1-carboxylate
N-{[7-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(pyrrolidin-1-yl)acetamide
N-methyl-2-(1,2,3,4-tetrahydroisoquinolin-5-yl)-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
1-(2,2-dimethylpropyl)-4-{[5-(trifluoromethyl)pyridin-2-yl]amino}pyrrolidin-2-one
N,2-dimethyl-N-[1-(pyridin-3-yl)pentyl]imidazo[1,2-a]pyridine-6-carboxamide
1-cyclopropyl-N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
[1-(isoquinolin-5-ylmethyl)-4-(2-phenylethyl)piperidin-4-yl]methanol
ethyl 4-[6-(5-fluoro-1H-indole-2-carbonyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
2-ethyl-5-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]-2H-1,2,3,4-tetrazole
3-butyl-1-methyl-4-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazin-2-one
N-[(2R,3R)-1'-[(2-fluoro-4-methoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-2-carboxamide
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methylfuran-2-yl)methyl]acetamide
N-(2,4-dimethylphenyl)-N'-methyl-N'-[1-(pyridin-2-yl)propan-2-yl]ethanediamide
4-[(3,4-dichlorophenyl)methyl]-2-(morpholin-4-ylmethyl)-1,4-oxazepane
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl){[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}amine
3-(carbamoylamino)-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]propanamide
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-(thiolan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-{2-[(pyridin-3-yl)amino]ethyl}propanamide
[1-(1-ethyl-1H-pyrazole-4-carbonyl)-3-[(2-methylphenyl)methyl]piperidin-3-yl]methanol
2-chloro-N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-4-fluoro-N-methylbenzamide
{3-[3-cyclopropyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]-5-methyl-1,2-oxazol-4-yl}methanol
N-ethyl-3-(3-hydroxy-3-methylbutyl)-N-propylbenzamide
1-(2-methoxyethyl)-4-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}piperazine
1-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-2-(2-methoxyethoxy)ethan-1-one
1-({5-[1-(5-fluoropyridin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)-4-methylpiperazine
N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-2-(methylsulfanyl)-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-chloro-3-methyl-N-[(2-phenoxypyridin-3-yl)methyl]benzamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(3-methyloxetan-3-yl)methyl]-1H-pyrazole-3-carboxamide
[(3R,5R)-5-[(dimethylamino)methyl]-1-[3-(3-methoxyphenyl)benzoyl]piperidin-3-yl]methanol
(3S,4R)-1-(1H-imidazol-4-ylmethyl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3-(pyrrolidine-1-sulfonyl)benzamide
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
3-[5-({[2-(2,6-dimethylphenoxy)ethyl](ethyl)amino}methyl)thiophen-2-yl]prop-2-yn-1-ol
2-cyclopropyl-4-methyl-5-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}pyrimidine
1-(1-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)pyrrolidin-2-one
5-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]-N-(propan-2-yl)pyrimidin-2-amine
[(2,6-difluoro-4-methoxyphenyl)methyl](methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
2-methyl-1-[1-(2-methyl-1-benzofuran-7-carbonyl)azetidin-3-yl]piperidine
1-(2-cyclopentylacetyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
1-[3-(furan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one