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N-[(3-chlorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
4-{5-fluoro-2-[4-(1H-pyrazol-5-yl)phenyl]pyrimidin-4-yl}morpholine
2-(4-{[4-(azepan-1-yl)quinazolin-2-yl]methyl}piperazin-1-yl)phenol
N-methyl-4-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)benzene-1-sulfonamide
N-(pyridin-3-ylmethyl)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-amine
2-[4-cyclopentyl-1-(3-methylbutyl)piperazin-2-yl]ethan-1-ol
6-[4-(2-methoxyethoxy)piperidin-1-yl]-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-[2,2-dimethyl-3-(4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazin-1-yl)propyl]morpholine
2-cyclopropyl-8-(1H-indol-5-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(piperidin-1-yl)-1-[4-(piperidin-3-yl)benzoyl]piperidine
4-{2,7-diazaspiro[4.5]decane-7-carbonyl}-N-(pyridin-4-ylmethyl)aniline
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
N-(3-benzylphenyl)-4-(2-methoxyethoxy)piperidine-1-carboxamide
(4aS,8aR)-6-(pyridazine-3-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-(3-fluoro-4-methoxybenzoyl)-1-[1-(furan-2-ylmethyl)piperidin-4-yl]piperidine
1-[2-(3,4-dimethoxyphenyl)ethyl]-5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)pyrrolidin-2-one
(4-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
2-{5-[morpholin-4-yl(phenyl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-(morpholin-4-yl)ethan-1-one
3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]propan-1-one
(4-{[methyl(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amino]methyl}oxan-4-yl)methanol
2-(4-fluorophenoxymethyl)-4-hydroxy-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]pyrimidine-5-carboxamide
1-{4-[(2-hydroxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(3-methoxyphenyl)ethan-1-one
N-[(2-chlorophenyl)methyl]-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-(propan-2-yl)acetamide
1-(3-phenylpropyl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
3-(4-benzyl-1H-pyrazol-5-yl)-1-(1H-pyrrole-2-carbonyl)piperidine
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-3,6-dimethyl-1-benzofuran-2-carboxamide
N-cycloheptyl-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
1-(2-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}ethyl)-4-(furan-2-carbonyl)piperazine
N-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methylcyclohexanamine
N-[(3R,4S)-1-(6-cyclopropylpyrimidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
N-(2-methoxyethyl)-1-[1-(2-methylpyridine-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(2-methylphenyl)ethyl]piperidine-3-carboxamide
methyl 6-[(2-fluorophenyl)methyl]-2-[(oxolan-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-fluoro-2-[1-(thiophene-3-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
N-cyclopentyl-4-[2-(3-fluorophenyl)-3-oxopiperazin-1-yl]-4-oxobutanamide
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[3-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methanol
methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl][(2-methyl-1H-imidazol-4-yl)methyl]amine
(2S)-1-{[7-fluoro-2-(4-methylphenyl)quinolin-3-yl]methyl}pyrrolidine-2-carboxamide
1-[2-(cyclohexylmethyl)morpholine-4-carbonyl]cyclopropane-1-carboxamide
N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-2-(2,3,6-trimethylphenoxy)acetamide
5-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
3-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-N-(1-phenylethyl)propanamide
3-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}-N,N-dimethyl-1,2,4-oxadiazole-5-carboxamide
3-{[(4-chlorophenyl)methyl]({[2-(propan-2-yl)pyrimidin-4-yl]methyl})amino}propan-1-ol
N-cyclohexyl-N-methyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
5-[(2E)-but-2-en-1-yl]-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,3,4-oxadiazole-2-carboxamide
(1S,5R)-6-benzyl-3-(4-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 5-{[(3,5-difluorophenyl)methyl]amino}-3-acetamido-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-1-ethyl-1H-1,2,4-triazole