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(3R,4R)-1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
methyl 5-[(3,3-dimethylcyclohexyl)amino]-3-acetamido-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[2-({3-azaspiro[5.5]undecan-9-yl}amino)ethyl]-4-fluorobenzamide
7-(cyclohexylmethyl)-2-[2-(1H-pyrazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
9-(2-methoxyethyl)-1-methyl-4-(3-phenylpropyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamide
1-ethyl-4-{[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-3,5-dimethyl-1H-pyrazole
N-(1,2-oxazol-5-ylmethyl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
N-cyclopentyl-2-({2-[(3-methylpyridin-2-yl)amino]ethyl}amino)propanamide
2-({2-amino-3-ethyl-3H-imidazo[4,5-b]pyridin-6-yl}formamido)-N-(propan-2-yl)acetamide
2-acetyl-8-[4-methyl-6-(methylamino)pyrimidin-2-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(cyclohexylmethyl)-N-(1H-imidazol-4-ylmethyl)piperidin-3-amine
N-{4-[3-(dimethylamino)piperidine-1-carbonyl]phenyl}ethane-1-sulfonamide
2-hydroxy-3-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
1-(3-methoxyphenyl)-4-(2-methyl-2-phenylpropanoyl)piperazin-2-one
1-(4-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
8-(3,5-dimethylbenzoyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
8-(5-methyl-2H-1,2,3-triazole-4-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(dimethylamino)-N-ethyl-2-(4-methylphenyl)-N-(oxan-4-ylmethyl)acetamide
[3-(prop-2-en-1-yl)-1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]methanol
(3aS,6aS)-2-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(2-methylpropanesulfonyl)ethyl]-4-(2-oxopyrrolidin-1-yl)benzamide
N3-[3-(dimethylamino)-2,2-dimethylpropyl]-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3-({1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}methyl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
6-cyclopentyl-3-{[(4,6-dimethylpyrimidin-2-yl)amino]methyl}-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(furan-2-yl)ethane-1,2-dione
5-(4-methoxypiperidine-1-carbonyl)-2-(3-phenylpropyl)-1,3-benzoxazole
4-{1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-4-yl}pyrimidin-2-amine
N-[(1-ethyl-1H-indazol-3-yl)methyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
ethyl 4-[5-(4-methoxyphenyl)-1,2,4-triazin-3-yl]piperazine-1-carboxylate
1-(1-acetylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
ethyl 4-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
(3aS,6aS)-2-cyclopentanecarbonyl-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(2-methylprop-2-en-1-yl)oxy]-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
{1-[5-(cyclobutylamino)-5,6,7,8-tetrahydroquinazolin-2-yl]piperidin-4-yl}methanol
3-{[3-(3-phenylphenyl)-1H-pyrazol-1-yl]methyl}pyridine
3-cyclohexyl-N-{2-[4-(4-methyl-1,4-diazepane-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}propanamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-amine
(1-{3-[(4-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidin-4-yl)(pyridin-2-yl)methanol
1-methyl-2-({3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)piperidine
2-cyclopropyl-9-[2-(methylsulfanyl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
3-cyclohexyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-4-carboxamide
N-{4-[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]-2-methoxyphenyl}acetamide
1-(2-{[6-(dimethylamino)pyrimidin-4-yl]amino}ethyl)piperidine-3-carboxamide
3-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-3-methyl-1-[3-(2-methylphenyl)phenyl]urea
6-[2-(phenylamino)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(2S,4R)-1-[(3,4-difluorophenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}pyrrolidine-2-carboxamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]propane-1-sulfonamide
2-[3-(2-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-methylpyrimidine