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4-(2-methyl-1H-imidazol-1-yl)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidine-4-carboxylic acid
(3aS,6aR)-5-[(2-fluorophenyl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(2R,3R)-3-(dimethylamino)-1'-[(4-ethoxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-3-(5-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-({1-[(2-aminopyridin-3-yl)methyl]piperidin-3-yl}methyl)-2-(4-methoxyphenyl)acetamide
N-[2-(benzylsulfanyl)ethyl]-2-(pyrrolidin-1-yl)pyrimidine-5-carboxamide
N-[(1-ethyl-1H-indazol-3-yl)methyl]-3-phenyl-1H-pyrazole-4-carboxamide
4-acetamido-N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]butanamide
4-{1-cyclohexyl-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazol-3-yl}pyridine
6-(5-methyl-1H-indole-2-carbonyl)-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
4-(4-chlorophenyl)-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]butanamide
2-(3-methoxypropyl)-3-oxo-N-[2-(propan-2-yl)phenyl]-2,8-diazaspiro[4.5]decane-8-carboxamide
N-({3-methyl-7-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(phenylsulfanyl)acetamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2,6-difluorobenzene-1-sulfonamide
ethyl 1-[(4-methoxyphenyl)methyl]-5-(oxolane-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-{1-[2-(diethylamino)ethyl]-1H-imidazol-2-yl}-7-fluoro-1,2-dihydroquinolin-2-one
2-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-3-yl}-1H-1,3-benzodiazole
6-(2-chlorophenyl)-N-(2-ethoxyethyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(pyridin-4-yl)-4-[4-(pyrrolidin-1-ylmethyl)benzoyl]piperazine
N-{[2-(3-hydroxypiperidin-1-yl)-7-methylquinolin-3-yl]methyl}-2-oxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2,3-dimethylquinoxaline-6-carboxamide
ethyl 2-[7-(2,5-difluorobenzoyl)-2,7-diazaspiro[4.5]decan-2-yl]acetate
N-methyl-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(1,3-thiazol-2-ylmethyl)pyridin-2-amine
N-{[2-(2-acetamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methylbenzamide
2-cyclopentyl-8-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 3-[(3S,4R)-4-(dimethylamino)-1-[(4-fluorophenyl)methyl]piperidin-3-yl]propanoate
N-[(2R)-2-hydroxypropyl]-5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carboxamide
2-[4-({[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]amino}methyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
2-methyl-N-(1,3-thiazol-2-yl)-3-(4H-1,2,4-triazol-4-yl)benzamide
N-[(1-ethylpyrrolidin-3-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-2-sulfonamide
1-[1,3-dioxo-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N,N-diethylpiperidine-4-carboxamide
1-(8-chloro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]urea
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-propylpyridine-4-carboxamide
(2S,4S)-N-ethyl-1-[2-(propan-2-yloxy)acetyl]-4-[2-(pyridin-4-yl)acetamido]pyrrolidine-2-carboxamide
4-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-oxobutanamide
N-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}cyclopropanamine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-N-(pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]octan-3-amine
4-(hydroxymethyl)-1-{[2-(methylsulfanyl)phenyl]methyl}azepan-4-ol
(2S)-4-methyl-2-{4-[1-(propan-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-1-yl}pentanamide
5-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(3-hydroxy-1,2-oxazol-5-yl)-N-(isoquinolin-5-ylmethyl)-N-methylpropanamide
3-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-1,3-oxazolidin-2-one
1-[3-({[2-(pyrazin-2-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-[1-(cyclohexylmethyl)piperidin-3-yl]-5-methyl-1,3-oxazole-4-carboxamide
1-[3-(4H-1,2,4-triazol-4-yl)benzamido]cyclopentane-1-carboxylic acid
1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
3-{[(5-fluoro-2-methylphenyl)methyl]amino}-1-(3-methylpiperidin-1-yl)propan-1-one
N-{2-[5-methyl-4-({2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamido}methyl)-1,3-oxazol-2-yl]phenyl}pyridine-3-carboxamide