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(1S,5R)-3-(2-methoxypyridine-3-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-(2,3-dihydro-1H-inden-5-yl)propanamide
6-(propan-2-yl)-2-(2-{[4-(propan-2-yl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
1-{[(3,5,7-trimethyl-1H-indol-2-yl)formamido]methyl}cyclopentane-1-carboxylic acid
1-[2-(dimethylamino)ethyl]-4-ethyl-3-[1-(pyridazine-3-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{[6-(2,3-dimethoxyphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}morpholine
3-({[7-(methylsulfanyl)-2-{[3-(trifluoromethyl)phenyl]methoxy}quinolin-3-yl]methyl}amino)-1λ6-thiolane-1,1-dione
2-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-3,4,7-trimethyl-1H-indole
2-[2-(3-methylbut-2-en-1-yl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
N-cyclopropyl-1-{1-[2-(methylsulfanyl)benzoyl]piperidin-4-yl}piperidine-4-carboxamide
N-({7-[3-(1H-indol-3-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
1-[2-(4-methoxyphenyl)ethyl]-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-benzyl-5-(4-ethylpiperazin-1-yl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[1-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-4-yl)-2-(3-methoxyphenyl)ethyl]-N-methylfuran-2-carboxamide
N-ethyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-(pyridin-4-ylmethyl)acetamide
4-{1-[3-(4-fluorophenyl)benzoyl]piperidin-4-yl}-2-phenylpyrimidine
N-(cyclopropylmethyl)-1-[1,3-dioxo-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-propylpiperidine-3-carboxamide
(4S,4aS,8aS)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-phenyl-decahydroquinolin-4-ol
N-[2-(pyrrolidin-1-yl)ethyl]-2-{4-[2-(thiophen-3-yl)acetyl]morpholin-3-yl}acetamide
3-[2-(dimethylamino)ethyl]-5-[1-(4-fluorobenzoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
1-(4-ethoxy-3-methylphenyl)-4-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]butane-1,4-dione
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
3-(1-ethyl-1H-imidazol-2-yl)-1-{[4-(trifluoromethyl)phenyl]methyl}piperidine
4-(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)-2,1,3-benzoxadiazole
4-cyclobutyl-2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-methylpyrimidine
N3-butyl-1-(furan-2-ylmethyl)-4-oxo-N5-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
4-(dimethyl-1,2-oxazol-4-yl)-3-[1-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-3-(3-methoxy-4-methylphenyl)propan-1-one
3-(piperidin-4-ylmethyl)-6-propyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
6-(azepan-1-yl)-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-[(ethanesulfonyl)methyl]-7-(4-fluorophenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(4-fluorophenyl)methyl]piperazin-2-one
(3S,4S)-4-(propan-2-yloxy)-1-(5-propyl-1,3,4-oxadiazole-2-carbonyl)pyrrolidin-3-ol
3-(3-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl)propanoic acid
N-cyclohexyl-1-methyl-2-oxo-6-(propan-2-yl)-N-(thiophen-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[3-(pyridin-2-yl)propyl]pyridin-2-amine
N-[(5-chloro-2-methoxyphenyl)methyl]-2-(3,4-dimethoxyphenyl)-N-ethylacetamide
(2S,4S,5R)-1-methyl-2-(2-methylpropyl)-5-(pyridin-3-yl)-4-{[(1r,4r)-4-hydroxycyclohexyl]carbamoyl}pyrrolidine-2-carboxylic acid
1-(2,6-dimethylquinoline-3-carbonyl)-N-ethylpyrrolidine-3-carboxamide
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
2-methyl-1-(3-{[(2-methylhexan-3-yl)amino]methyl}piperidin-1-yl)propan-1-one
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-{[(3S,4S)-3-hydroxy-4-(3-methoxyphenyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
3-tert-butyl-1-methyl-4-[(1E)-1-phenylprop-1-en-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4,4-difluoro-1-({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)piperidine
(1S,5R)-3-cyclobutanecarbonyl-6-(3-phenylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
{3-[(3-methoxyphenyl)methyl]-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl}methanol
N-methyl-4-[(2-methylpyridin-3-yl)oxy]-N-[(3-methylthiophen-2-yl)methyl]piperidine-4-carboxamide