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N-methyl-3-{2-methyl-2,8-diazaspiro[4.5]decane-8-carbonyl}pyridin-2-amine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methyl-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-(2-{[1-(pyrazin-2-yl)propan-2-yl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-ethyl-5-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
[(3S,5R)-1-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
5-(2,4-dimethoxyphenyl)-N-[(3-methylpyridin-4-yl)methyl]-1,2,4-triazin-3-amine
7-fluoro-3-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,2-dihydroquinolin-2-one
N-[4-({[3-(pyrrolidin-1-yl)propyl]carbamoyl}methyl)phenyl]butanamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[3-(pyridin-3-yl)propyl]acetamide
2-(4-hydroxy-4-phenylpiperidin-1-yl)-2-[3-(methylcarbamoyl)phenyl]acetic acid
3-{imidazo[1,2-a]pyridin-2-yl}-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)propanamide
6-methoxy-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3,3-dimethyl-1-[(5-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea
1-methyl-3-[4-(4-{[(5-methylthiophen-2-yl)methyl]amino}piperidin-1-yl)phenyl]imidazolidin-2-one
5-phenyl-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1,2-oxazole-4-carboxamide
1-(4-fluorophenyl)-4-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)piperazine
1-{2-[1-(7-fluoro-3-methyl-1H-indole-2-carbonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
[2-(1H-imidazol-1-yl)ethyl](methyl)[(5-propylfuran-2-yl)methyl]amine
3,5-dimethyl-4-[1-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)pyrrolidin-2-yl]-1,2-oxazole
2-(3-fluorophenyl)-1-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}ethan-1-one
1-(1,3-benzothiazol-2-ylmethyl)-4-ethyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-N,5-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-[(2-phenyl-1,3-thiazol-4-yl)methyl]urea
5-{1-[(5-methoxy-1H-indol-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}pyrimidin-2-amine
3-methyl-1-[4-(2-methylbutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]butan-1-ol
methyl 5-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
ethyl 3-[(2-fluorophenyl)methyl]-1-(thiophene-2-carbonyl)piperidine-3-carboxylate
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepane-1-carboxamide
2-(3,5-difluorophenyl)-N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]acetamide
7-chloro-2-[(2-methyl-4-phenylpiperazin-1-yl)methyl]-4-(morpholin-4-yl)quinazoline
2-{4-methyl-6-[3-(1H-pyrazol-3-yl)phenyl]pyrimidin-2-yl}phenol
2-(2-methoxyethyl)-9-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-(2-oxo-2-{4-[4-(propan-2-yl)-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}ethyl)imidazolidin-2-one
5-{1-[(3-fluoro-4-methylphenyl)methyl]-1H-imidazol-2-yl}-2-methoxypyrimidine
[(1,2-dimethyl-1H-indol-3-yl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
1-{2-[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]-2-oxoethyl}-1,2-dihydroquinolin-2-one
3-methyl-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
N-[2-(morpholin-4-yl)ethyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
[(2-methoxyphenyl)methyl](pyridin-2-ylmethyl)(pyridin-3-ylmethyl)amine
N-(5-acetyl-2-ethoxyphenyl)-4-(3-oxo-3,4-dihydropyrazin-2-yl)piperazine-1-carboxamide
1,3,6-trimethyl-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)(pyridin-2-ylmethyl)amine
N-benzyl-2-(3-chloro-4-hydroxyphenyl)-N-(3-hydroxy-2-methylpropyl)acetamide
N-(oxan-4-yl)-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
1,3-dimethyl-5-(2-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(1H-pyrazol-1-yl)propan-1-one
7-chloro-4-[(2-ethylpyrimidin-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-5-fluoro-1H-1,3-benzodiazole
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]acetamide