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4-[5-({[(4,6-dimethylpyridin-2-yl)methyl](methyl)amino}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
4-(1H-1,3-benzodiazole-2-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
2-(3-fluorophenyl)-1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
1-[(3-methoxyphenyl)methyl]-4-({4-[(3-methoxypropyl)amino]-6-methylquinazolin-2-yl}methyl)piperazin-2-one
4-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-2-amine
N-[4-(4-{[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]-N-(1-phenylcyclopropyl)acetamide
3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]-4-[(4-phenylphenyl)methyl]piperazin-2-one
N,N-dimethyl-5-{[(4-methylphenyl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(3-fluoropyridin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
N-cyclopropyl-1-[1-(3,3-dimethylbutanoyl)piperidin-4-yl]piperidine-3-carboxamide
1-{[3-cyclopropyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}piperidine
N-cyclopropyl-5-[(isoquinolin-5-yloxy)methyl]-N-(2-methylpropyl)-1,2-oxazole-3-carboxamide
1-[2-(3-fluorophenyl)piperidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl)methyl]acetamide
methyl 3-[2-(4-methoxyphenyl)acetyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-methyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
N-({7-[(2,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
3-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}-6-methyl-1,2-dihydroquinolin-2-one
[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-2-yl]methanol
methyl({3-[(1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-yl)oxy]phenyl}methyl)(thiophen-3-ylmethyl)amine
6-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]pyridine-2-carbonitrile
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-(4-hydroxypiperidin-1-yl)-N-methylacetamide
N-cyclopropyl-1-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
N4-[(1-ethyl-1H-imidazol-2-yl)methyl]-N4,N6,N6-trimethylpyrimidine-4,6-diamine
(2S)-2-(1H-1,2,3,4-tetrazol-1-yl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
4-[4-oxo-7-(oxolan-3-ylmethyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-4-phenylbenzamide
7-(3-phenylpropyl)-2-(pyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-(4-methyl-1,3-thiazol-5-yl)-1-[2-(2-phenylethyl)morpholin-4-yl]propan-1-one
2-{imidazo[1,2-a]pyridin-3-yl}-1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}ethan-1-one
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}azepane-1-sulfonamide
ethyl 3-[(2-methylphenyl)methyl]-1-(1,2-oxazol-3-ylmethyl)piperidine-3-carboxylate
5-{1-[(2E)-3-(3,4-difluorophenyl)prop-2-enoyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
5-{1-[(2-hydroxyphenyl)methyl]piperidin-4-yl}-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
2-(1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)acetamide
N-butyl-1,5,6-trimethyl-N-[(3-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N,5-dimethyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
ethyl 2-[4-(2,1,3-benzothiadiazol-4-ylmethyl)piperazin-1-yl]pyridine-3-carboxylate
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-(thiophen-2-ylmethyl)piperidine
4-(cyclopropylamino)-5-methyl-N-(3-methylbutyl)thieno[2,3-d]pyrimidine-6-carboxamide
3-cyclohexyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1H-pyrazole-4-carboxamide
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-2-(1,3-thiazol-4-yl)acetamide
1-{2-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-{[methyl(2-phenylethyl)amino]methyl}-2-oxo-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,2-dihydropyridine-3-carboxamide
7-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)-N-methyl-N-(thian-4-yl)acetamide
N-[2-(1H-imidazol-4-yl)ethyl]-4-(piperidin-3-yl)benzamide