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(3S,4R)-N,N-dimethyl-4-propyl-1-{thieno[3,2-d]pyrimidin-4-yl}pyrrolidin-3-amine
(3S,4R)-1-[(2-aminopyridin-3-yl)methyl]-4-(2,3-dimethoxyphenyl)pyrrolidine-3-carboxylic acid
8-(1-ethyl-5-oxopyrrolidine-3-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl[(2-phenyl-1,3-thiazol-4-yl)methyl]{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(3S,4R)-1-(8-methoxy-4-methylquinolin-2-yl)-4-propylpyrrolidin-3-yl]acetamide
diethyl({[3-(2-propylpyrrolidine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
1-{3-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
1-(3-methylbutyl)-3-(2-methylpropyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methyl-9-(5-methyl-1,3-oxazole-4-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
methyl (2S,4S,5R)-1,2-dimethyl-4-[methyl(1,2-oxazol-3-ylmethyl)carbamoyl]-5-(2-methylphenyl)pyrrolidine-2-carboxylate
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dimethoxybenzamide
1-methyl-2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-indole
N-{[5-methyl-2-(4-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}cyclopentanecarboxamide
1-{2-methyl-5-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]phenyl}imidazolidin-2-one
ethyl 4-[(1-cycloheptyl-5-oxopyrrolidin-3-yl)amino]piperidine-1-carboxylate
8-(3,4-diethoxybenzoyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
ethyl 1-[(4-methoxyphenyl)carbamoyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
4-(2-fluoro-3-methoxyphenyl)-5,6-dimethyl-2-(trifluoromethyl)pyrimidine
4-(2-hydroxy-4-methoxybenzoyl)-5-methyl-1-(3-methylphenyl)piperazin-2-one
5-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-2-(morpholin-4-ylmethyl)-4H-pyran-4-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(2-phenylacetyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-{[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]amino}ethyl)pyridine-4-carboxamide
1-(2-phenylethyl)-5-(1,3-thiazol-4-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
5-{1-[(4-methoxynaphthalen-1-yl)methyl]piperidin-4-yl}-5-(3-methylbutyl)imidazolidine-2,4-dione
6-(aminomethyl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]pyrimidin-4-amine
(2S,4R)-1-[(2-chlorophenyl)methyl]-N,N-diethyl-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
methyl 4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
1-[(2-methylpyrimidin-5-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[(4-methylphenyl)methyl]benzamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,3-dimethyl-5,6-dihydro-1,4-dioxine-2-carboxamide
methyl (2S,4S,5R)-4-[(2,2-dimethylpropyl)carbamoyl]-1,2-dimethyl-5-(2-methylphenyl)pyrrolidine-2-carboxylate
2-(4-{[(5-ethylpyrimidin-2-yl)amino]methyl}piperidin-1-yl)ethan-1-ol
1-methyl-3-(propan-2-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}-1H-pyrazole-5-carboxamide
1-[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-4-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-1,2,3-triazole
1-(6-fluoro-4-methylquinazolin-2-yl)-N-[(3-fluorophenyl)methyl]azepan-4-amine
1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-3-(3-methoxypropyl)piperidine
2-[(2-fluorophenyl)methyl]-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-1,6-dimethyl-1,4-dihydropyridin-4-one
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
2-[(1H-imidazol-2-ylmethyl)(pyridin-2-ylmethyl)amino]butan-1-ol
2-(ethanesulfonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
5-ethyl-2-methyl-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]pyrimidin-4-amine
2-{5-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1H-pyrazol-3-yl}pyridine
3-(4-methyl-1,3-thiazol-5-yl)-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]amine
(3aS,6aS)-5-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-1-oxo-2-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
methyl[2-methyl-2-(morpholin-4-ylmethyl)propyl](oxan-2-ylmethyl)amine
1-[2-amino-6-(cyclopropylamino)pyrimidin-4-yl]-4-(piperidin-1-yl)piperidine-4-carboxamide
[(4,5-dimethylfuran-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one