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1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
methyl 3-acetamido-5-{[(4-acetamidophenyl)methyl]amino}-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-N-phenylpyrimidin-2-amine
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-3-(1H-imidazol-1-yl)propan-1-one
2-{[(4-fluorophenyl)methyl](methyl)amino}-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
4-(4-methyl-1H-pyrazol-1-yl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidine-4-carboxylic acid
3-(2,4-difluorophenyl)-1-(pyridin-2-ylmethyl)-6-(1,3-thiazole-4-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-(methoxymethyl)-6-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pyrimidine
2-(1-benzofuran-2-yl)-2-(thiomorpholin-4-yl)acetic acid
N-(adamantan-2-yl)-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
N-({3-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-(2,5-dioxoimidazolidin-4-yl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]acetamide
3-(3-hydroxy-3-methylbutyl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}benzamide
2-(2,3-dihydro-1-benzofuran-7-ylformamido)-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
6-(2-chlorophenyl)-N-[(5-methylfuran-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-cyclopropyl-N-methyl-6-oxo-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,6-dihydropyrimidine-5-carboxamide
N-(1H-indol-2-ylmethyl)-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2S)-N-ethyl-1-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]pyrrolidine-2-carboxamide
3-{1-[5-(1,3-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-3-methylbutyl}pyridine
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(pyridin-2-yl)ethyl]acetamide
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]ethan-1-one
2-(2-{[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]methyl}phenoxy)ethan-1-ol
2-acetyl-N-(2-methoxyethyl)-N-[(4-methylphenyl)methyl]benzamide
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-4-(morpholin-4-yl)benzamide
2-[2-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,2,3,4-tetrahydrophthalazine-1,4-dione
(3R,4R)-4-(morpholin-4-yl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-ol
methyl 2-(1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-[(3S,4R)-3-acetamido-4-(4-methylphenyl)pyrrolidin-1-yl]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
2-ethyl-5-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
3-[(dimethylamino)methyl]-1-[2-(4-fluorophenoxy)ethyl]piperidin-3-ol
6-{[4-(dimethylamino)oxan-4-yl]methyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-[2-oxo-2-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)ethyl]-1,3-oxazolidin-2-one
4-{1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidin-3-yl}benzoic acid
ethyl 3-[(2-methylphenyl)methyl]-1-(thiophene-3-sulfonyl)piperidine-3-carboxylate
[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]({[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
N-ethyl-2-(2-methanesulfonylacetamido)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
3-(5-methylthiophen-2-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
(4aS,8aR)-1-(3-methoxypropyl)-6-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-decahydro-1,6-naphthyridin-2-one
N-[(3S,4R)-1-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1-methyl-4-[(6-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridin-3-yl)methyl]piperazine
2-{2-benzyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-1,3-thiazole-4-carboxamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]-1,3-thiazole
2-(cyclopent-2-en-1-yl)-N-[1-(morpholin-4-ylmethyl)cyclopentyl]acetamide
4-[(2,3,6-trifluorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
5-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
{1-[(8-methoxy-2H-chromen-3-yl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
N-(2,5-dihydroxy-2-methylpentyl)-3-methyl-1H-indole-2-carboxamide