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N-(3-methylphenyl)-3-{1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidin-4-yl}propanamide
(4-benzyl-1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)methanol
[(3R,4R)-4-[(dimethylamino)methyl]-1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methanol
1-ethyl-3-methyl-N-{[4-(methylsulfanyl)phenyl]methyl}-N-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
2-{2-[(4-ethyl-3-oxopiperazin-1-yl)methyl]-4-(thiophen-2-yl)phenoxy}acetic acid
N,3,6-trimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-benzofuran-2-carboxamide
5-{1-[2-(2-methylphenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
(1R,7S)-3-[4-(2-hydroxyethyl)phenyl]-N-(1H-imidazol-2-ylmethyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-butyl-4-(5-methyl-1,3-oxazole-4-carbonyl)-1-(3-phenylphenyl)piperazin-2-one
N-[2-(4-phenyl-4H-1,2,4-triazol-3-yl)ethyl]aniline
1-[(2-butyl-1H-imidazol-4-yl)methyl]-N-[3-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl]propan-1-ol
2-[2-({3-azaspiro[5.5]undecan-9-yl}amino)ethyl]-5,6-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
(4S)-3,3,4-trimethyl-1-(1,3-thiazole-4-carbonyl)piperidin-4-ol
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(1-propylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
N-(1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
(1S,5R)-6-[(3-chloro-2-fluorophenyl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-{1-[(2-ethoxyphenyl)methyl]-4-[(6-ethoxyquinolin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]quinoxaline
4-[1-(9H-purin-6-yl)piperidin-4-yl]piperazin-2-one
3-chloro-4-methyl-N-(1,4-oxazepan-6-ylmethyl)benzene-1-sulfonamide
4-[7-(2-methoxypyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
2-(furan-2-ylmethyl)-9-(5-oxopyrrolidine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-chloro-2-[(1E)-2-methyl-3-{methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}prop-1-en-1-yl]phenol
1-{[1-butyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-3-ol
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(1H-indol-2-ylmethyl)methylamine
9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-{[4-(2-methylpropyl)phenyl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(2-acetylphenyl)pyrazine-2-carbonitrile
5-{[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]methyl}-2-methoxybenzoic acid
3-methyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-1H-pyrazole-5-carboxamide
3-(piperidine-1-carbonyl)-5-[4-(propan-2-yl)piperazin-1-yl]-1-propyl-4,5,6,7-tetrahydro-1H-indazole
[5-({4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)-2-(propan-2-yloxy)phenyl]methanol
(4aR,7aS)-1-benzyl-4-(2-cyclopropylacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methoxy-4-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1,3-thiazole-5-carboxamide
methyl({[5-(oxan-2-yl)furan-2-yl]methyl}){[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}amine
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)thiophene-2-sulfonamide
2-(1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
1-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1H-imidazole-2-carboxamide
3-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,2,5-trimethyl-1H-pyrrole
8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
N-[1-ethyl-2-(3-methoxyphenyl)-7-(3-methoxypiperidine-1-carbonyl)-1H-1,3-benzodiazol-5-yl]acetamide
8-fluoro-3-(oxan-2-ylmethyl)-3,4-dihydroquinazolin-4-one
7-cyclohexyl-2-(5-ethyl-1,3,4-thiadiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-methoxy-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-[2-({1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)ethyl]piperidine-3-carboxamide
ethyl 1-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)-4-oxopiperidine-3-carboxylate
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-1H-pyrazole-4-carboxamide
2-(5-fluoropyridine-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one