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2-{8-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
1-(cyclohexylmethyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[(thiophen-2-ylmethyl)amino]methyl}piperidin-2-one
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[1-(2-phenoxypropanoyl)piperidin-4-yl]imidazolidine-2,4-dione
5-(2-phenylphenyl)furan-2-carboxamide
2-[1-(2-phenylethyl)-4-[6-(trifluoromethyl)pyridin-2-yl]piperazin-2-yl]ethan-1-ol
1-(4-{[3-(4-phenylbenzoyl)piperidin-1-yl]sulfonyl}phenyl)ethan-1-one
1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-amine
6-fluoro-4-methyl-2-{2-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]pyrrolidin-1-yl}quinazoline
3-(benzylamino)-N-[2-(1H-imidazol-1-yl)ethyl]-5-(phenylsulfamoyl)benzamide
N-[(2-chlorophenyl)methyl]-3-[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]propanamide
8-[3-(3-chlorophenyl)propanoyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(3aR,5R,6S,7aS)-2-{[2-(2-phenylethoxy)phenyl]methyl}-octahydro-1H-isoindole-5,6-diol
N-methyl-3-(3-{[(2,2,2-trifluoroethyl)carbamoyl]amino}phenyl)propanamide
N-[(3R,4S)-1-(1-aminocyclopropanecarbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-5-propylpyrimidin-4-amine
N-(2-methoxyethyl)-3-(2-methoxyphenyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]propanamide
3-[4-(3-chlorophenyl)piperazine-1-carbonyl]-2-(cyclopentylmethyl)-1,6-dimethyl-1,4-dihydropyridin-4-one
(3S)-N,N-dimethyl-1-[2-(pyrrolidin-1-yl)benzoyl]azepan-3-amine
N-{3-[ethyl(phenyl)carbamoyl]phenyl}oxolane-3-carboxamide
(1S,6R)-3-[3-(2-methoxyphenyl)benzoyl]-3,9-diazabicyclo[4.2.1]nonane
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
[(5-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1,3,4-oxadiazol-2-yl)methyl]dimethylamine
3-[(4-methylpiperazin-1-yl)sulfonyl]-5-phenyl-N-(pyridin-3-ylmethyl)benzamide
N-(4-{[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]carbamoyl}-2-methylphenyl)furan-2-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-1-{4-[(1-methylpiperidin-4-yl)methyl]piperazin-1-yl}ethan-1-one
N-cyclopropyl-N-[(4-hydroxy-3-methoxyphenyl)methyl]-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
dimethyl[3-(2-{[(2S)-4-methyl-2-phenylpiperazin-1-yl]methyl}phenoxy)propyl]amine
1-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-3-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]urea
N-{2-[methyl(phenyl)amino]ethyl}oxane-2-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-4-methyl-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
(2S,4R)-4-amino-N-ethyl-1-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)pyrrolidine-2-carboxamide
1-(2-methylphenyl)-4-{1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}piperazine
1-(oxolane-2-carbonyl)-4-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperazine
4-({4-methyl-5-[1-(6-methylpyrimidin-4-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
4-(1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrrolidin-3-yl)-2-(pyridin-4-yl)pyridine
2-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]acetic acid
(2S)-4-methyl-1-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]-2-(propan-2-yl)piperazine
1-methyl-N-[2-(pyridin-2-yl)ethyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-ethyl-4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-(propan-2-yl)piperazine
3-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrazolo[1,5-a]pyrimidine
5-(1H-imidazol-2-yl)-1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-phenyl-1H-imidazole
propyl (2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate
(3R,4S)-4-cyclopropyl-N,N-dimethyl-1-(pyridine-4-carbonyl)pyrrolidin-3-amine
(4aR,8aR)-2-(3-hydroxypyridine-2-carbonyl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(2,3,6-trimethylphenoxy)acetamide
4-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}morpholine
6-(2,4-dimethoxyphenyl)-N,N-dimethylpyrazin-2-amine