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2-(1-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-1H-imidazol-2-yl)quinoline
7-(cyclobutylmethyl)-N-(2-methylphenyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
N-(1-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-7-fluoroquinazolin-4-amine
1-(2-phenylethyl)-5-[2-(piperidin-1-yl)acetyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-cyclohexyl-N-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)piperazine-1-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]propan-1-one
6-(2H-1,3-benzodioxole-5-carbonyl)-1-(cyclopropylmethyl)-3-(2,3-dimethoxyphenyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(2S,4R)-N-ethyl-1-(2-methylpropyl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
5-(3-methoxy-2-methylphenoxymethyl)-3-(phenoxymethyl)-1,2,4-oxadiazole
5-{3-[3-(4-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
1-cyclohexyl-6-(pyridin-2-ylmethoxy)-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
1-(dimethyl-1,3-oxazole-4-carbonyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
benzyl(methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
2-(4-methylbenzoyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
3-ethyl-1-methyl-N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)-1H-pyrazole-5-carboxamide
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)acetamide
N-methyl-2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-methyl-6-oxo-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
3-hydroxy-1-(2-methoxyethyl)-3-(thiomorpholin-4-ylmethyl)piperidin-2-one
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
6,7-dimethoxy-2-(1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
5-(morpholin-4-ylmethyl)-N-(naphthalen-1-ylmethyl)-1,2-oxazole-3-carboxamide
1-{6-[3-(4-fluorophenyl)pyrrolidin-1-yl]pyrimidin-4-yl}piperidin-4-ol
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}[1-(pyridin-3-yl)propan-2-yl]amine
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-7-methoxy-1,2,3,4-tetrahydronaphthalen-2-amine
2-[2-({4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]pyridine
(3S,4R)-4-(3-fluorophenyl)-1-(1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)pyrrolidine-3-carboxylic acid
2-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-5-methoxypyridin-4-ol
2-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
2-[(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-5-methylpyrazine
4-(hydroxymethyl)-5-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,2-oxazole-3-carboxamide
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
N-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-(pyridin-3-ylmethyl)piperidin-4-amine
2-{1,4-bis[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[4-(4-{[7-chloro-4-(morpholin-4-yl)quinazolin-2-yl]methyl}piperazin-1-yl)phenyl]ethan-1-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)furan-3-carboxamide
ethyl 4-[(2-chlorophenyl)methyl]-1-(4-oxo-4-phenylbutanoyl)piperidine-4-carboxylate
(1S,5R)-6-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentan-1-one
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-dimethylpiperidin-4-amine
(4aS,7aR)-1-(1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-3-{methyl[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propanamide
N-[cyclopropyl(pyridin-2-yl)methyl]-N,2,6,8-tetramethylquinoline-4-carboxamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
N-methyl-N-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}oxolan-3-amine
2-(adamantan-1-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide