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2-methoxy-1-{1'-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
N-[2-fluoro-6-(trifluoromethyl)phenyl]-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
3-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(1H-pyrazol-4-yl)phenyl]urea
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(naphthalen-1-ylmethyl)propanamide
3-cyclopropyl-1-[2-(dimethylamino)-4-(4-hydroxypiperidin-1-yl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{3-[6-(piperazin-1-yl)pyridin-2-yl]phenyl}acetamide
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-2-(pyridin-3-yl)pyridine
N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyrazin-2-ylmethyl)acetamide
7-(1,3-benzothiazol-2-yl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[(2-chlorophenyl)methyl]-1-[(2E)-4-methylpent-2-en-1-yl]-1,4-diazepan-5-one
2-(4-fluorophenyl)-N-methyl-N-(piperidin-4-yl)imidazo[1,2-a]pyridine-6-carboxamide
7-(4-fluorophenyl)-2-[(5-methylfuran-2-yl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(4-fluorophenyl)piperazine
3-methoxy-6-(6-methoxypyridin-3-yl)pyridazine
N,2-dimethyl-N-(naphthalen-1-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
1-cyclopropyl-6-oxo-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-3-carboxamide
1-(cyclopropylmethyl)-5-[1-(2-methylpropyl)-5-oxopyrrolidine-3-carbonyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(3,4-dimethylphenyl)-3-(3-methoxyphenoxy)azetidine-1-carboxamide
N-(1-cycloheptylpiperidin-3-yl)but-3-enamide
[3-(1H-indol-1-yl)propyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
1-ethyl-4,6-dimethyl-3-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-1,2-dihydropyridin-2-one
4-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)quinoline
methyl 1-[2-hydroxy-3-(3-{[(3-methoxypropyl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
3-methyl-8-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N,2-dimethyl-6-(propan-2-yl)pyrimidin-4-amine
(4aS,8aR)-6-(3-ethoxypropanoyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
7-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2-oxa-7-azaspiro[4.5]decane
(1S,5R)-6-benzyl-3-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(4-fluorophenyl)methyl]-1-(2-{[(2-hydroxy-3-methoxyphenyl)methyl]amino}ethyl)-1H-1,2,3-triazole-4-carboxamide
N-[2-(2-fluorophenoxy)pyridin-3-yl]-4-methyl-1,4-diazepane-1-carboxamide
(benzylsulfamoyl)(methyl){2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}amine
2-{4-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
1-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-4-propylpiperazine
2-amino-4-(1,2-dimethyl-1H-imidazol-5-yl)-6-(1H-indol-3-yl)pyridine-3-carbonitrile
N-[(2-chloropyridin-3-yl)methyl]-5-[(3-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N-({3-methyl-7-[3-(prop-2-en-1-yloxy)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-sulfonamide
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-(2-fluorophenoxy)azetidine
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[(3-methylphenyl)methyl]piperidine
6-{[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
2-methyl-6-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]pyrimidin-4-ol
1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-4-(1H-pyrazol-4-yl)butan-1-one
(4aS,8aS)-2-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-decahydro-2,7-naphthyridin-4a-ol
N-[(2S,4R,6S)-2-ethyl-6-(1-ethyl-1H-pyrazol-4-yl)oxan-4-yl]acetamide
[(3R,5R)-1-(2-aminopyridine-4-carbonyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
1-(2-methoxy-5-{[(oxan-4-ylmethyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
1-{2-hydroxy-3-[4-methoxy-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
1-{2-[6-hydroxy-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepan-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
(3S,4R)-1-(2-chloro-6-fluoro-3-methylbenzoyl)-4-phenylpyrrolidine-3-carboxylic acid