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(4-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}-1,4-oxazepan-6-yl)methanol
1,2-dimethyl-3-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-1H-indol-5-ol
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine-1-carboxamide
5-[2-(4-fluorophenyl)azetidine-1-carbonyl]-2,4-dimethyl-1,3-thiazole
9-{2-[4-(methylsulfanyl)phenyl]acetyl}-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
8-benzyl-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2R,3R)-1'-[(2E)-3-(4-fluorophenyl)prop-2-enoyl]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
N-{3-[5-(trifluoromethyl)pyridin-2-yl]propyl}methanesulfonamide
N-(1,3-benzothiazol-2-yl)-3-[2-(pyridin-3-yl)piperidin-1-yl]propanamide
3-(1-benzothiophen-7-yl)-6-(2-cyclopropylacetyl)-1-(cyclopropylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(3R,4R)-3-cyclopropyl-1-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-4-methylpyrrolidin-3-ol
8-[2-(5-chloro-6-methyl-1-benzofuran-3-yl)acetyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
1-(2-chlorophenyl)-3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]urea
[(3S,5R)-1-(3-fluoropyridine-2-carbonyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
5-cyclohexanecarbonyl-1-(cyclopropylmethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[3-(thiophen-2-yl)propanoyl]pyrrolidine-3-carboxylic acid
(3S,4S)-1-(benzenesulfonyl)-4-[4-(pyridin-4-yl)piperidin-1-yl]pyrrolidin-3-ol
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(1-methyl-3-phenyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[({2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)methyl]-3,4-dihydroquinazolin-4-one
1-[(3-methoxyphenyl)methyl]-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[3-(1H-pyrazol-3-yl)piperidin-1-yl]ethan-1-one
5-(2-chloroprop-2-en-1-yl)-7-({[2-(morpholin-4-yl)ethyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
4-(1-benzothiophen-2-ylmethyl)-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
({[2-(azocan-1-yl)pyridin-3-yl]methyl}sulfamoyl)dimethylamine
7-(cyclobutylmethyl)-2-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
2-methoxy-1-[1'-(3-phenylbutyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-(2-{2-[5-(hydroxymethyl)furan-2-yl]-1H-imidazol-1-yl}ethyl)pyridine-3-carboxamide
2-({2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}amino)-1,3-thiazole-4-carboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-(pyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[3-(2,5-difluorobenzoyl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
3-(but-2-yn-1-yl)-5-[1-(3-phenylbutyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
(1S,5R)-3-(3-chlorobenzoyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-2-ylmethyl)amine
N-ethyl-3-(1H-pyrazol-1-yl)-N-(pyridin-4-ylmethyl)benzamide
1-(3,5-dichloropyridin-2-yl)-4-hydroxypiperidine-4-carboxylic acid
7-chloro-4-[1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-methyl-2-[4-(2-phenoxyethyl)phenyl]propanamide
2-(furan-2-yl)-N-(4-methyl-2-oxo-1,2-dihydroquinolin-7-yl)azepane-1-carboxamide
4-({2-[3-(azepan-1-yl)-2-hydroxypropoxy]-5-chlorophenyl}methyl)piperazin-2-one
N-[(3S,4S)-4-methoxy-1,1-dioxo-1λ6-thiolan-3-yl]-2-[3-(trifluoromethyl)phenyl]acetamide
1-benzyl-N3-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(2-fluorophenyl)-2-[2-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)-4-phenylphenoxy]acetamide
1-methyl-4-[(3-methylquinoxalin-2-yl)methyl]-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
(2-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-oxoethyl)urea
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-fluoro-N-(pyridin-3-ylmethyl)benzamide
4-benzyl-1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-ethyl-1,4-diazepan-5-one
1-(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)piperidine-3-carboxamide
N-{[3-(3-methylbutyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]acetamide