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ethyl 4-[1-(cyclopent-3-en-1-yl)-4-phenyl-1H-imidazol-5-yl]-1H-pyrazole-3-carboxylate
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-methyl-N-[2-(morpholin-4-yl)ethyl]benzamide
2-[3-benzyl-1-(4-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-cyclobutylacetamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
1-cyclohexyl-6-(pyridin-2-ylmethoxy)-4-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,3-benzothiazole-5-carboxamide
(3S,4R)-1-[3-(methylsulfanyl)propyl]-4-phenylpyrrolidine-3-carboxylic acid
1-methyl-5-[(2-methylpropyl)amino]-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-methyl-6-[2-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
(2S,4R)-4-amino-1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-N-methylpyrrolidine-2-carboxamide
4-{2-[3-fluoro-5-(trifluoromethyl)phenyl]pyridine-4-carbonyl}morpholine
7-(2-methylphenyl)-9-(oxolan-3-yloxy)-4-[4-(trifluoromethyl)benzenesulfonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(4-hydroxyphenyl)-2-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]acetic acid
5-(3-{4-azatricyclo[4.3.1.13,8]undecan-4-yl}-3-oxopropyl)-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
5-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]-N-ethylpyrimidin-2-amine
1-(2-chlorophenyl)-3-(1-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
[(3R,4S)-1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(2-methyl-1H-indol-3-yl)ethan-1-one
1-(2H-1,3-benzodioxol-5-yl)-3-(2-phenylethyl)-5-[(propan-2-yloxy)methyl]-1H-1,2,4-triazole
1-(3,5-dimethylphenyl)-4-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperazin-2-one
1-(furan-2-ylmethyl)-3-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]urea
3-{imidazo[1,2-a]pyridin-2-yl}-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,2,4-oxadiazole
1-[(3S,4S)-3-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-4-hydroxypyrrolidin-1-yl]-2-(1H-imidazol-1-yl)ethan-1-one
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
2-{3-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
N-[3-({methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
4-[(2-fluorophenyl)methyl]-1-[3-(furan-2-yl)benzoyl]-1,4-diazepan-5-one
N-(1-benzylpyrrolidin-3-yl)-3-[1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]propanamide
N-(2-{7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
3-{2-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-1,3-thiazolidine-2,4-dione
7-(1-benzoxepine-4-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(2-methylpropyl)-6-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-butyl-3-[(4-fluorophenyl)formamido]-N-(pyridin-3-ylmethyl)propanamide
N-(2-phenylethyl)-N-(propan-2-yl)oxolane-3-carboxamide
(2S,3S)-3-methyl-2-({5-[(4-methylpiperazin-1-yl)methyl]furan-2-yl}formamido)pentanamide
2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-4-carboxamide
9-(2,6-dimethylpyridine-4-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
ethyl 1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidine-4-carboxylate
2-[4-(2-methoxyphenoxy)piperidin-1-yl]pyrazine
2-amino-4-[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]-6-(4-hydroxyphenyl)pyridine-3-carbonitrile
1-{1-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
methyl 3-({4-[3-(aminomethyl)pyrrolidin-1-yl]-6-oxo-1,6-dihydropyridazin-1-yl}methyl)-4-methoxybenzoate
2-methyl-4-[4-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)phenyl]but-3-yn-2-ol
2-[3-({4-ethyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)phenoxy]acetamide
N,6-dimethyl-N-{[2-(2-methylpropoxy)phenyl]methyl}-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[(3-chlorophenyl)methyl]-3-{1-[(2-hydroxy-6-methoxyphenyl)methyl]piperidin-4-yl}propanamide
2-(pyrrolidin-3-yl)-N-(quinolin-8-yl)benzamide
1-{4-[(3-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}-1,2-oxazol-5-yl)methoxy]phenyl}ethan-1-one
1'-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(5-methylpyridine-2-carbonyl)pyrrolidin-3-yl]methanol