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6-({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
(3S,4S)-1-[4-(piperidin-1-ylmethyl)benzoyl]-4-propylpyrrolidine-3-carboxylic acid
3-({2-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]acetamido}methyl)-4-methylbenzoic acid
2-methoxy-3-{1-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-imidazol-2-yl}quinoline
1-[(2-phenyl-1H-imidazol-4-yl)methyl]-4-(thiophen-2-ylmethyl)piperazine
4-{1-[(2-ethoxyphenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
4-{[(1-methyl-1H-pyrazol-4-yl)methyl]sulfamoyl}-N-[(3S)-pyrrolidin-3-yl]benzamide
3-[(dimethylamino)methyl]-3-hydroxy-N-(2-phenoxyphenyl)piperidine-1-carboxamide
9-[(3-methoxyphenyl)methyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1,4-dioxan-2-ylmethyl)-N-methyl-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
6-(2-fluoro-5-methoxyphenyl)-N2,N2-dimethylpyrimidine-2,4-diamine
4-chloro-2-[(1E)-3-[4-(5-fluoropyrimidin-2-yl)piperazin-1-yl]-2-methylprop-1-en-1-yl]phenol
3-fluoro-4-(6-hydroxyhexyl)benzene-1-sulfonamide
4-[4-(4-chlorophenoxy)piperidine-1-carbonyl]pyridin-2-amine
1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-4-phenylpiperidine-4-carbonitrile
(2S)-N-cyclopropyl-2-acetamido-N-{[4-(methylsulfanyl)phenyl]methyl}pentanediamide
5-(2-cyanophenyl)-N-propylthiophene-2-carboxamide
7-(1,3-benzothiazol-2-yl)-4-(1H-indol-2-ylmethyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})(pyridin-3-ylmethyl)amine
8-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
7-(cyclopropylmethyl)-2-(pyrrolidine-1-carbonyl)-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]ethan-1-one
[1-(adamantan-2-yl)-4-[(2-chlorophenyl)methyl]piperidin-4-yl]methanol
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-4-hydroxy-N-methyl-2-(thiophen-2-yl)pyrimidine-5-carboxamide
N-[cyclohexyl(thiophen-2-yl)methyl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-1-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
2-[cyclohexyl(methyl)amino]-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}pyridine-3-carboxamide
2-(3-{[(2-hydroxyethyl)[(1-methyl-1H-imidazol-2-yl)methyl]amino]methyl}phenyl)-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[1-(pyridin-3-yl)propan-2-yl]benzamide
5-(hydroxymethyl)-2-methyl-4-{[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}pyridin-3-ol
(3S,4S)-4-methyl-1-(9H-purin-6-yl)piperidine-3,4-diol
3-[(dimethylamino)methyl]-N-(3-acetamido-4-fluorophenyl)-3-hydroxypiperidine-1-carboxamide
N,2,5,7-tetramethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]quinoline-4-carboxamide
2-methyl-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-1-(oxolan-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indol-4-one
1-methyl-3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-indole
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanamide
(4aR,8aS)-6-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]methylamine
2-{[(1S,5R)-6-[(dimethylcarbamoyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzoic acid
(2E)-3-(3-fluorophenyl)-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}prop-2-enamide
1-[2-(benzyloxy)ethyl]-4-(1H-pyrrole-3-carbonyl)-1,4-diazepan-6-ol
5-(furan-2-yl)-3-({2-[5-(oxan-2-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)-1,2-oxazole
N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)-2-(pyridin-2-yl)acetamide
N-{[1-({3-[4-(methoxymethyl)-6-oxo-1,6-dihydropyrimidin-2-yl]phenyl}methyl)piperidin-3-yl]methyl}acetamide
N-[(1-benzyl-4-phenylpiperidin-4-yl)methyl]-2-(1-methyl-3-oxopiperazin-2-yl)acetamide
1-(2-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-2-methyl-1H-imidazole
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-4-[(3-methylphenyl)sulfanyl]piperidine
N-[3-(dimethylamino)-2,2-dimethylpropyl]-5-methyl-4-{[1-(thiophen-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
1-(furan-2-carbonyl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-1,4-diazepane