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2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-1-phenoxypropan-2-ol
N-({1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}methyl)pyridine-3-carboxamide
3-{[(4-benzyl-5-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}pyridine
1-(1-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-3-phenylpropan-1-ol
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-(2-phenyl-1H-imidazol-1-yl)acetamide
2-(dimethylamino)-2-(4-methylphenyl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
(2S)-N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methylcyclopropanecarbonyl)piperidine
5-(methoxymethyl)-N-[(3-methoxyphenyl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-benzyl-1-[4-(thiophen-2-yl)butanoyl]-1,4-diazepan-5-one
N-[1-(4-methoxyphenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(1H-1,2,4-triazol-1-yl)acetamide
1-(4-{4-[3-(diethylamino)pyrrolidine-1-carbonyl]phenoxy}piperidin-1-yl)-2-methoxyethan-1-one
(1-methyl-1H-imidazol-2-yl)(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)methanol
1-[(1R,2S)-2-(methoxymethyl)cyclopentyl]-2-[2-(trifluoromethyl)phenyl]-1H-imidazole
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]propan-1-ol
8-(dimethyl-1,3-oxazole-5-carbonyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(3S)-1-{[5-(2-ethoxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3-fluoropyrrolidine
{1-[(1-pentylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-methyl-6-(piperidin-3-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrimidin-4-amine
3-({2-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
4-[(6-methylpyridin-3-yl)oxy]-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
{5-methyl-3-[4-(2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-1,2-oxazol-4-yl}methanol
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-3-(2-oxoazepan-1-yl)propanamide
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
ethyl 2-cyclohexyl-3-oxo-3-{5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}propanoate
5-{[furan-2-yl(phenyl)methyl]carbamoyl}-1H-imidazole-4-carboxylic acid
1-(pyridin-3-ylmethyl)-4-[(4-{[1-(thiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine
1-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]cyclopropane-1-carboxamide
4-[2-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]pyrimidin-2-amine
1-cycloheptyl-N-(3-hydroxy-2,2-dimethylpropyl)-6-oxopiperidine-3-carboxamide
methyl 4-(3-{[(3,5-dimethoxyphenyl)formamido]methyl}piperidin-1-yl)-4-oxobutanoate
[4-(oxan-2-ylmethyl)-1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl]methanol
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-methylurea
4-{[(butan-2-yl)[(4-methylphenyl)methyl]amino]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(3-methoxypropyl)-1H-pyrazole-4-carboxamide
N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-{[3-(2-aminoethyl)phenyl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
dimethyl({2-[3-(4-phenylphenyl)-1,2,4-oxadiazol-5-yl]ethyl})amine
1-cyclopropyl-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
5-(3-{2-azabicyclo[2.2.1]heptan-2-yl}-3-oxopropyl)-5-(thiophen-2-ylmethyl)pyrrolidin-2-one
2,2-difluoro-N-({1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)butanamide
4-{4-[(3-chloro-4-methoxyphenyl)methyl]-2-oxopiperazin-1-yl}benzonitrile
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-4-phenylpiperidine-4-carboxamide
4-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2,5-dimethylpyrimidine
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-(5-fluoro-2-methyl-1H-indol-3-yl)ethan-1-one
4-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)azetidin-3-yl]pyridine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,4-dimethyl-1,3-thiazole-5-carboxamide
2-(2-methoxyphenyl)-1-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazole