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1-(1-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-benzyl-3-[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-N-methylpropanamide
4-methoxy-N-methyl-3-(1H-pyrazol-4-yl)benzamide
6-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-(pyridin-4-ylmethyl)acetamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-4-(1H-pyrazol-5-yl)benzamide
N-{[7-chloro-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)oxolane-2-carboxamide
2-(2,3-dimethylphenyl)-4-{1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}pyridine
1-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
(3aR,6aR)-2-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-1,3-benzodiazole
(1R,2S,4R)-N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
4-[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)carbamoyl]pyridin-1-ium-1-olate
1'-[(3-chloro-2-fluorophenyl)methyl]-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(4-methoxyphenyl)-N-[4-(4-{[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
2-chloro-5-acetamido-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]benzamide
N-[(2-fluorophenyl)methyl]-3-{1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]piperidin-3-yl}propanamide
5-({4-[(3-chlorophenyl)methyl]piperazin-1-yl}methyl)isoquinoline
1-tert-butyl-4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyrrolidin-2-one
2-(2-methoxyethyl)-9-(2-phenoxypropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(1H-1,2,3,4-tetrazol-5-yloxy)-N-[(2,3,5-trifluorophenyl)methyl]aniline
4-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-1-phenyl-1H-1,2,3-triazole
1,3-dimethyl-5-({[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(2,5-difluorophenyl)methyl]-1-(4,7-dimethylquinazolin-2-yl)piperidine-4-carboxamide
N-methyl-5-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
3-({[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)benzonitrile
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2,3-dimethyl-1H-indole-7-carboxamide
4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-[(3-methoxyphenyl)methyl]morpholine
(4aR,7aS)-1-propanoyl-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-1-{[5-(4-chlorophenyl)furan-2-yl]methyl}-N-(2-phenylethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
N,2-dimethyl-N-[1-(pyridin-3-yl)propyl]-1-benzofuran-5-carboxamide
N-cyclohexyl-N-[(4-methoxy-2,5-dimethylphenyl)methyl]-3-methyl-1,2-oxazole-5-carboxamide
1-{3,9-diazaspiro[5.5]undecan-3-yl}-2-(morpholin-4-yl)ethane-1,2-dione
2-(3-methoxypropyl)-9-[2-(2-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-4-hydroxy-3-methoxybenzamide
5-cyclohexaneamido-1-(2-methoxyethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
3-chloro-5-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,2-dihydropyridin-2-one
{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
(2R,6S)-1-(1-ethyl-1H-pyrazole-3-carbonyl)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
(2S)-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-hydroxy-3-phenylpropan-1-one
N-cyclopropyl-2-ethoxy-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
8-[2-(3-chlorophenyl)-2-hydroxyacetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{2-[5-(1-cyclopropanecarbonylpiperidin-2-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}morpholine
(3aR,6aR)-N-ethyl-2-methyl-N-(oxan-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(5-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-methyl-1H-pyrazole-5-carboxamide
N-[(dimethyl-1,3-oxazol-4-yl)methyl]-3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide