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methyl 2-(3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamido)-4-(methylsulfanyl)butanoate
3-(cyclopropylmethyl)-1-[4-(1H-imidazol-1-yl)benzoyl]piperidine-3-carboxylic acid
N-cyclopentyl-N-{[4-(oxolan-3-yloxy)phenyl]methyl}-3-phenyl-1H-pyrazole-5-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
(2H-1,3-benzodioxol-5-ylmethyl)({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
1-[3-(4-{2-[3-({methyl[(5-oxopyrrolidin-2-yl)methyl]amino}methyl)phenoxy]ethyl}piperazine-1-carbonyl)phenyl]pyrrolidin-2-one
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]acetamide
N-ethyl-2-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]furan-3-carboxamide
2-({4-[2-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
2-methyl-N-[2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)propyl]-1,3-thiazole-4-carboxamide
N-{1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}pyridin-2-amine
methyl 7-oxo-3-(quinolin-7-ylmethyl)-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(2-{2-[3-(furan-2-yl)phenyl]-1H-imidazol-1-yl}ethyl)pyrazine
N-(furan-3-ylmethyl)-N-methyl-5-propyl-1,2-oxazole-3-carboxamide
N-(3-ethoxypropyl)-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
6-(cyclohex-3-ene-1-carbonyl)-1-(cyclopropylmethyl)-3-(2-methylquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-(3-methyl-1,2-oxazol-5-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
2-(4-chloro-1-methyl-1H-pyrazol-3-yl)-1H-1,3-benzodiazole-6-carboxylic acid
1-[(4aS,8aR)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-2-methoxyethan-1-one
(1S,4S)-2-(2,5-dimethoxyphenyl)-5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
1-[(4,6-dimethylpyrimidin-2-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
{5-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]furan-2-yl}methanol
5-[(4-chloro-3-methyl-1H-pyrazol-1-yl)methyl]-3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]pyrrolidin-3-yl]methanol
4-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-1-(4-methylphenyl)piperazin-2-one
3-(2H-1,3-benzodioxol-5-yl)-1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]propan-1-one
5-methoxy-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,3-dimethyl-1H-indole-2-carboxamide
4-[2-(2-chlorophenyl)ethyl]-11-{[2-(propan-2-yloxy)ethyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
5-methyl-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)acetamide
2-[(1S,5R)-6-(benzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
2-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}-1-(piperidin-1-yl)ethan-1-one
1-methyl-4-phenyl-3-[1-(pyridin-4-ylmethyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]acetamide
2-{[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]amino}-N-(pyrazin-2-yl)acetamide
3-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-N-[(3,4-difluorophenyl)methyl]propanamide
3-(2H-1,3-benzodioxol-5-yl)-5-[5-(methoxymethyl)furan-2-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-methyl-2-(1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
N-benzyl-N-methyl-3-{1-[2-(pyridin-4-yl)acetyl]piperidin-4-yl}propanamide
N-[2-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)propyl]-2H-1,3-benzodioxole-5-carboxamide
5-(methoxymethyl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}furan-2-carboxamide
2-[(2-chlorophenyl)methyl]-4-[5-(methoxymethyl)furan-2-carbonyl]morpholine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-[2-(butan-2-yl)phenoxy]acetamide
3-(oxolan-3-yl)-5-{3-[4-(propan-2-yl)phenyl]propyl}-1,2,4-oxadiazole
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-3-(pyridin-3-yl)propan-1-one
6-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}pyrimidin-4-ol
methyl[2-(4-methylphenoxy)ethyl]{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
5-[4-hydroxy-1-(thiophen-3-ylmethyl)piperidin-4-yl]-N-(2-methoxyphenyl)-1-benzofuran-2-carboxamide
1-{2-[(cyclopentylamino)methyl]-5-methoxyphenoxy}-3-(pyrrolidin-1-yl)propan-2-ol
[(3R,5R)-1-(2-cyclopropylpyrimidine-5-carbonyl)-5-[(dimethylamino)methyl]piperidin-3-yl]methanol