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methyl (2S)-1-[3-(1H-indole-2-carbonyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]pyrrolidine-2-carboxylate
2-{4-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]morpholin-2-yl}ethan-1-amine
2-{1-[(3,4-difluorophenyl)methyl]-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
(3R,4S)-4-[ethyl({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)amino]oxolan-3-ol
1-{[methyl({[3-(methylsulfanyl)phenyl]methyl})carbamoyl]methyl}piperidine-4-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,4-dimethyl-1H-imidazole-2-carboxamide
2-chloro-N-{2-[(4-methyl-1H-imidazol-5-yl)formamido]ethyl}benzamide
1-[3-(4-methylbenzenesulfonamido)propyl]-3-(1,2,3-thiadiazol-5-yl)urea
5-(3,3-diphenylpiperidine-1-carbonyl)-1-methyl-1H-pyrrole-3-carbonitrile
1-methyl-4-(pyridin-3-ylmethyl)-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]propan-1-one
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
2-[methyl(phenyl)amino]-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(cyclohex-1-en-1-yl)-1-{2-[5-(morpholine-4-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}ethan-1-one
1-cycloheptyl-6-oxo-N-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-3-carboxamide
N-[4-chloro-3-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]carbamoyl}amino)phenyl]-2-methoxyacetamide
(3S,4R)-4-(2-methylphenyl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}pyrrolidine-3-carboxylic acid
2-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}thiophene-3-sulfonamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(methylamino)-N-(pyridin-3-ylmethyl)pyridine-4-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
2-[4-(6-chloro-1,3-benzothiazol-2-yl)-1H-pyrazol-1-yl]-N-(1-ethyl-1H-1,2,3-triazol-4-yl)acetamide
N-[(2R,3R)-2-(benzyloxy)-1'-(pyrazine-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
4-({5-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)morpholine
3-(4-hydroxybutyl)-6-methyl-5-phenyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-{4-[4-(morpholin-4-yl)piperidine-1-carbonyl]phenyl}ethane-1-sulfonamide
4-(3,6-dimethylpyrazin-2-yl)-2-(6-methoxynaphthalen-2-yl)morpholine
1-{2-[({imidazo[1,2-a]pyridin-3-ylmethyl}amino)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
4-methoxy-N-(2-methoxyethyl)-2-{[1-(1,3-oxazole-5-carbonyl)piperidin-4-yl]oxy}benzamide
2-{[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3-methylpyridine
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(propan-2-yl)acetamide
2-methyl-N-[1-({[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]furan-3-carboxamide
7-(cyclobutylmethyl)-2-(1H-1,2,4-triazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
8-[(3-chloro-2,6-difluorophenyl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6,8-dimethyl-4-(piperidine-1-carbonyl)-2-(pyrimidin-5-yl)quinoline
1-(furan-2-ylmethyl)-N-[(4-sulfamoylphenyl)methyl]piperidine-3-carboxamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-methanesulfonamidopropanamide
2-(2,5-dimethylphenyl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
2-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-dihydrophthalazin-1-one
3-(3,4-dimethyl-1H-pyrazol-5-yl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}propanamide
9-(2,3-dihydroxybenzoyl)-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-ethyl-9-(1-methyl-1H-pyrazole-4-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
2-(2-{[4-(6-methylpyridin-2-yl)piperazin-1-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
5-chloro-3-methyl-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1H-indole-2-carboxamide
6-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
1-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]-6-oxopiperidine-3-carboxamide
3-[(2,3-dichloro-6-fluorophenyl)methyl]-1,3-oxazolidin-2-one
2-[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-6-methylpyridine-3-carboxylic acid
3-(2-methoxyphenyl)-5-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetamide
N-cyclopentyl-1-(2-methylpropyl)-5-(1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide