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3-{[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]methyl}-N-methyl-1,2,4-oxadiazole-5-carboxamide
N-(furan-3-ylmethyl)-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)-1,8-naphthyridine-2-carboxamide
8-(6-aminopyridine-3-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
8-[1-(3-chloro-4-methylphenyl)piperidin-4-yl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
3-(azepane-1-sulfonyl)-5-(6-methoxypyridin-3-yl)benzoic acid
N-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
2-amino-4-(3,5-dimethyl-1H-pyrazol-4-yl)-6-[4-(morpholin-4-yl)phenyl]pyridine-3-carbonitrile
2-[(3-methoxypiperidin-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
4-{imidazo[1,2-a]pyrimidine-2-carbonyl}-1-[(4-methoxyphenyl)methyl]piperazin-2-one
3-(4-chlorophenyl)-3-phenyl-N-[2-(pyrazin-2-yl)ethyl]propanamide
1-(3,4-difluorophenyl)-4-(1,2-oxazolidine-2-carbonyl)pyrrolidin-2-one
3-{2-[(2,4-dimethoxyphenyl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}phenol
(4aR,8aR)-7-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
N-[(5-chlorothiophen-2-yl)methyl]-5-propyl-1,3,4-oxadiazol-2-amine
4-cyclopentyl-2-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrimidine
1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[3-(dimethylamino)-2,2-dimethylpropyl]-1H-pyrazole-4-carboxamide
methyl 3-(7-chloro-2-{[(5-methyl-1H-pyrazol-3-yl)formamido]methyl}-2,3-dihydro-1-benzofuran-5-yl)benzoate
4-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-3-(3-fluorophenyl)piperazin-2-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-methanesulfonamidoacetamide
1-{2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(2-methoxyethoxy)piperidine
3-({[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]amino}methyl)-N,N-dimethylpyridin-2-amine
1-[(4-chlorophenyl)methyl]-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
N-[(5-chlorothiophen-2-yl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2S,4R)-4-amino-N-methyl-1-(4-propylpyrimidine-5-carbonyl)pyrrolidine-2-carboxamide
1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
2-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}-N-(1-methyl-1H-pyrazol-4-yl)acetamide
N-[(4-cyanophenyl)methyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
1-(oxan-4-yl)-4-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]piperidine
N-(2,3-dimethylquinoxalin-6-yl)-4-(pyrimidin-2-yl)-1,4-diazepane-1-carboxamide
3-{2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
methyl({2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})(3-phenylbutyl)amine
5-{[4-(piperidin-1-yl)butanamido]methyl}thiophene-2-carboxylic acid
4-methoxy-N-{1-[1-(1-phenoxypropan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-(cyclopropylmethyl)-4-methyl-5-{1-[2-(morpholin-4-yl)ethyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
N-cyclopropyl-5-(1-methylpiperidine-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(3R,4R)-1-(1-benzofuran-2-ylmethyl)-4-cyclobutyl-3-methylpiperidin-4-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-4-(1H-pyrazol-1-yl)benzamide
8-[2-(2,3-dimethylphenoxy)ethyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-1-[1-(pyrimidin-2-yl)piperidin-3-yl]urea
6-(2-methoxyphenyl)-N-(oxan-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N3-methyl-4-oxo-1-(3-phenylpropyl)-N5-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-1,4-dihydropyridine-3,5-dicarboxamide
1-(2,3-dimethylphenyl)-4-{[4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl]methyl}piperazine
(4aR,7aS)-1-acetyl-4-(2-oxo-4-phenylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[(1H-indol-4-ylmethyl)amino]-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
4-(1H-1,3-benzodiazol-1-yl)-1-(4-methoxypyrimidin-2-yl)piperidine-4-carboxylic acid
4-(5-methylpyridin-2-yl)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-4-ol
2-methoxy-N-(1-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide