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8-methoxy-2-methyl-4-{[4-(methylsulfanyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]acetamide
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-3-(1H-pyrazol-1-yl)benzamide
2-{2-[1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-2-yl]ethyl}pyridine
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[4-(trifluoromethyl)phenyl]ethan-1-one
1-[(2-fluorophenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
8-[(3-hydroxyphenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2-methoxyphenyl)methyl]-4-methyl-2-(4-methylpiperazin-1-yl)-N-(prop-2-en-1-yl)pyrimidine-5-carboxamide
3-{1-[4-(furan-2-yl)benzoyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[(5-methylhexan-2-yl)amino]adamantan-1-ol
2-(3-fluorophenyl)-N-(1-{4-[2-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)acetamide
4-(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)-3-(furan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-{1-[2-(morpholin-4-yl)benzoyl]piperidin-4-yl}piperidin-4-ol
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-(cyclohexylmethyl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(2S)-1-({3-[(dimethyl-1H-1,2,4-triazol-5-yl)carbamoyl]phenyl}methyl)pyrrolidine-2-carboxamide
3-(4-chlorophenyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-3-phenylpropanamide
3-(4-methyl-1,3-thiazol-5-yl)-N-[3-(4-methylbenzenesulfonamido)propyl]propanamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
N3-cycloheptyl-4-oxo-1-(propan-2-yl)-N5-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-benzyl-2-{6-oxo-2,7-diazaspiro[4.5]decan-2-yl}acetamide
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amine
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-(1,2-oxazol-3-ylmethyl)propanamide
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-4-methylpentan-1-one
N-[3-(3,6-dimethylpyrazin-2-yl)propyl]methanesulfonamide
2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]acetic acid
5-methyl-1-{2-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2S)-2-amino-4-hydroxy-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)butanamide
N-[2-(morpholin-4-yl)ethyl]-4-{4-[(quinolin-6-ylmethyl)amino]piperidin-1-yl}benzamide
3-(ethylsulfanyl)-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
3-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,5-dichlorophenyl)urea
1-[2-({[(5-fluoro-2-methylphenyl)methyl]amino}methyl)-5-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[2-(diethylamino)ethyl]-N-ethylpropanamide
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(quinazolin-4-yloxy)ethan-1-one
4-benzyl-1-(1,4-dioxan-2-ylmethyl)-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(1H-imidazol-2-yl)-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine
7,7-dimethyl-2-(morpholin-4-yl)-N-[(trimethylpyrazin-2-yl)methyl]-5,6,7,8-tetrahydroquinazolin-5-amine
3-(4-methyl-1,3-thiazol-5-yl)-1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}propan-1-one
(3R,4R)-1-{[5-(methoxymethyl)furan-2-yl]methyl}-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
6-methyl-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}imidazo[2,1-b][1,3]thiazole-5-carboxamide
1-[3-(2-chlorophenoxy)azetidin-1-yl]-3-(pyridin-3-yl)propan-1-one
(2R,6R)-1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
1-(6-chloro-1,3-benzothiazol-2-yl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-4-amine
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-methyl-N-(2-methylpropyl)piperidine-3-carboxamide
2-[methyl(2-phenylethyl)amino]-N-(oxan-3-yl)-2,3-dihydro-1H-indene-2-carboxamide
methyl 3-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-{4-[4-(4-methylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
6-(2H-1,3-benzodioxol-5-yl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one