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(3R,5S)-N-butyl-1-(pyridin-4-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
[(2S)-1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
1-(2-fluorophenyl)-N-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
4-(5-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
N-tert-butyl-2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoacetamide
3-[1-(oxan-4-ylmethyl)-1H-1,2,3-triazol-4-yl]benzonitrile
1-oxo-N-[(1R,2S)-2-phenylcyclopropyl]-1,2-dihydroisoquinoline-4-carboxamide
4-ethyl-3-(piperidin-3-yl)-1-[2-(1H-1,2,4-triazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2-fluorophenoxy)-N-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)azetidine-1-carboxamide
2-(4-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
5-(4-oxo-3,4-dihydrophthalazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(2R,6S)-2,6-dimethyl-4-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}morpholine
4-(4-fluorobenzenesulfonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
8-pentyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N3-cyclooctyl-N5-(3-ethoxypropyl)-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
9-(3-chloro-5-fluorobenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
3-[(cyclobutylamino)methyl]-1-[(3,4-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
8-benzyl-1-oxa-8-azaspiro[4.6]undecan-9-one
5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-one
3-amino-1-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}pyrrolidine-3-carboxylic acid
1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-4-(pyrrolidine-1-carbonyl)piperidine
3-[3-(2-chlorophenyl)pyrrolidin-1-yl]-5-(3-fluoro-4-methoxyphenyl)-1,2,4-triazine
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methylacetamide
{2-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-8-methylquinolin-3-yl}methanol
2-{4-cyclohexyl-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
(7S,9aR)-N-(3-fluorophenyl)-7,8-dimethyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
2,6-dimethoxy-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}benzamide
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-2-(2-oxopiperidin-1-yl)acetamide
8-methoxy-2-methyl-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 3-[4-(2-amino-3-cyano-5,6,7,8-tetrahydro-1,6-naphthyridin-4-yl)-1H-pyrazol-1-yl]propanoate
1-({4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-1,3-oxazol-2-yl}methyl)-1H-1,3-benzodiazole
4-[2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]-2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazole
4-[1-(carbamoylmethyl)-1H-imidazol-2-yl]-N-[(4-methylphenyl)methyl]piperidine-1-carboxamide
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole
2-ethyl-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2H-1,2,3,4-tetrazol-5-amine
N-[1-(morpholin-4-ylmethyl)cyclopentyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
N-[1-({4-[2-(3-methylpiperidin-1-yl)ethoxy]phenyl}methyl)piperidin-4-yl]acetamide
N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(furan-2-ylmethyl)propanamide
(4S,6R)-6-methyl-N-[3-(methylcarbamoyl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-sulfanylidene-1,3-diazinane-4-carboxamide
ethyl 1-(3-fluorobenzenesulfonyl)-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
4-methyl-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
N-[1-(1-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
(3R,5S)-1-benzyl-N-cyclooctyl-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrrolidin-3-amine
2-(1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2,3-dihydro-1H-indene-2-carbonyl}piperidin-4-yl)ethan-1-ol
methyl 5-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-3-acetamido-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[(4-fluorophenyl)methyl]-4-[5-(methoxymethyl)thiophene-2-carbonyl]-1,4-diazepane
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-methyl-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-{4-[(3-methylbutyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one