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N-[(3S,4R)-4-(4-methylphenyl)-1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-yl]acetamide
2-[(3R)-3-hydroxy-3-phenylpropyl]-1,2-dihydroisoquinolin-1-one
1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
ethyl 4-[(4-{[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
2-[4-(pyrimidin-2-yl)piperazin-1-yl]-1-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethan-1-one
6-chloro-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)pyridine-2-carboxamide
2-{[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
(4aR,8aS)-1-[2-(2-fluorophenyl)ethyl]-6-[(2-hydroxy-5-methoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-(piperazine-1-carbonyl)benzene-1-sulfonamide
2-methyl-6-({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)heptan-2-ol
N-(isoquinolin-5-ylmethyl)-1-(2-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-N-[(5-methylpyrazin-2-yl)methyl]piperidin-4-amine
3-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
5-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-3-phenyl-1,2-oxazole
8-(4-aminopyrimidin-2-yl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(dimethylamino)ethyl]-6-methyl-N-[(3-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-benzyl-8-[(2-hydroxyphenyl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-methoxy-4-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
2-(cyclobutylmethyl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(2S)-2-{[7-acetyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propanamide
dimethyl({4-methyl-5-[1-(naphthalen-2-ylmethyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
methyl 4-[4-(2-amino-6-methoxypyrimidin-4-yl)piperazin-1-yl]benzoate
5-[4-(diphenylmethyl)piperazin-1-yl]-1-(prop-2-yn-1-yl)azepan-2-one
8-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(adamantan-1-ylsulfanyl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]acetamide
7-[(4-fluoro-3-methoxyphenyl)methyl]-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N,N-dimethyl-3-[4-(4-methylphenoxy)piperidine-1-carbonyl]piperidine-1-carboxamide
N-[3-(3-carbamoylpiperidin-1-yl)propyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
3-(3-chlorophenyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-phenylpropanamide
N-(2-{7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
methyl 3-[2-(2-methoxyphenyl)acetyl]-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-amino-7-[1-methyl-3-(thiophen-2-yl)-1H-pyrazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-[2-(pyridin-2-yl)pyrrolidin-1-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
(1R,7S)-6-(piperidine-1-carbonyl)-3-[2-(pyridin-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
3-(4-{octahydropyrrolo[1,2-a]piperazin-2-yl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)pyridine
2-butyl-N-[(2-methylphenyl)(pyridin-4-yl)methyl]-1,3-benzoxazole-5-carboxamide
(E)-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-2-phenyl-N-(pyridin-2-ylmethyl)ethene-1-sulfonamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(pyridin-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(1S,5R)-3-benzoyl-6-(1-methyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(1H-indol-3-yl)-6-methylpyridine-3-carboxamide
4-[(2,3-dichlorophenyl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-(1H-pyrazol-3-ylmethyl)piperidine
3-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-fluorophenyl)urea
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methoxypyridine
N-{[8-(5-ethyl-1,3,4-oxadiazol-2-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}furan-2-carboxamide
(9-propyl-3-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-3,9-diazaspiro[5.5]undecan-1-yl)methanol
8-{[4-(4-chlorophenyl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
3-butyl-4-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-1-methylpiperazin-2-one
N-{2-[7-(quinolin-4-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-2-carboxamide
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-2-(pyridin-4-yl)acetamide