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4-(3,4-dimethoxyphenyl)-3-(3-methylthiophen-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(3,4,5-trimethoxyphenyl)-1H-imidazole
2-[(4-chlorophenyl)methyl]-4-{4-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
4-[(4-{4-[(2-methylphenyl)methyl]-2,5-dioxoimidazolidin-4-yl}piperidin-1-yl)methyl]-1H-pyrazole-3-carboxylic acid
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
8-[3-(1H-imidazol-1-yl)propyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methyl-N-(2-phenoxyphenyl)piperidine-1-carboxamide
2-(2-methoxyethyl)-4-{[3-(methylsulfanyl)phenyl]methyl}morpholine
1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-3-phenylpiperidine
4-methyl-5-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]-2-oxo-1,2-dihydropyridine-3-carbonitrile
1-(1H-imidazol-4-ylmethyl)-4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
5-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-4-ol
1-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
3-[4-(3-fluoropyridin-2-yl)piperazin-1-yl]propanamide
1-[(4aR,8aS)-6-(5-acetylthiophene-3-carbonyl)-decahydro-1,6-naphthyridin-1-yl]-2-(2-chloro-6-fluorophenyl)ethan-1-one
5-{4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
N-methyl-5-(morpholin-4-ylmethyl)-N-(thiophen-2-ylmethyl)-1,2-oxazole-3-carboxamide
(3R)-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3,4,4-trimethylpyrrolidin-3-ol
2-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-N-methylacetamide
N-[(3S,4R)-4-propyl-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl]methanesulfonamide
(1S,3R)-3-amino-N-{2-[(2-methyl-1H-imidazol-1-yl)methyl]phenyl}cyclopentane-1-carboxamide
{2-[2-(3,4-dimethoxyphenyl)phenoxy]ethyl}dimethylamine
[(1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl](methyl)amine
N-{7-[4-(methoxymethyl)piperidine-1-carbonyl]-1-methyl-2-phenyl-1H-1,3-benzodiazol-5-yl}ethane-1-sulfonamide
3-(3-methylbutyl)-8-[3-(pyridin-4-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-phenyl-N-{[7-(quinolin-4-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)piperidine-1-carboxamide
6-chloro-3-[(3-hydroxypiperidin-1-yl)methyl]-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-[2-(3-fluorophenyl)ethyl]-1-[(3-methylphenyl)methyl]pyrrolidine-2-carboxamide
N-(1-{7-[(4-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
2-(pyridin-3-ylmethyl)-9-(4,4,4-trifluorobutanoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-2-methyl-1-benzofuran-5-carboxamide
5-({[(3-{2-[4-(4-chlorobenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
9-(2-hydroxyacetyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(4-{2-[2-(3-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2-methylpropan-1-one
methyl 5-({5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}carbamoyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxylate
1-methyl-N-(3-methylbutyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{2-[(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
1-(adamantan-2-yl)-5-[2-(ethylamino)ethyl]pyrrolidin-2-one
2-(4-{[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]methyl}phenoxy)acetamide
1-(2-aminoethyl)-N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(4aS,7aR)-1-(3-ethyl-1H-indole-2-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-3-(3-chlorophenyl)-1-(cyclopropylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-{2-[2-(trifluoromethyl)phenyl]ethyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(3-methylphenyl)-2-{4-[3-(thiophen-3-yl)propanoyl]morpholin-3-yl}acetamide
(3S,5R)-1-(5-methylhexanoyl)-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid