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diethyl({4-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}methyl)amine
N,2,3-trimethyl-N-[(1-methylpiperidin-2-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(2-oxopyrrolidin-1-yl)acetamide
3-methoxy-N-(1-{7-[(4-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-hydroxyacetamide
4-(4-fluoro-2-{[2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzamide
2-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
(1R,5S)-8-(3,5-dichloro-4-methylbenzoyl)-3,8-diazabicyclo[3.2.1]octane
N,N-dimethyl-3-[2-(2-phenylethyl)morpholine-4-carbonyl]aniline
2-chloro-5-{1-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}pyridine
4-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[3-(2-oxopyrrolidin-1-yl)phenyl]piperazine-1-carboxamide
4-{[(2S)-2-benzyl-3-oxopiperazin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
1-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
(2S,4R)-4-amino-1-(pent-4-enoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-methoxy-N-[2-(5-methylfuran-2-yl)ethyl]-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
(3S,4S)-1-(4-methylbenzoyl)-4-(naphthalen-2-yl)piperidin-3-ol
2-(3-acetyl-1H-indol-1-yl)-N-methyl-N-(1H-pyrazol-5-ylmethyl)butanamide
3-(5-methyl-1H-pyrazol-1-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
6-[3-(3-fluorophenoxymethyl)piperidine-1-carbonyl]-2-(2-methoxyethyl)-1,3-benzoxazole
1-{6-hydroxy-4-[1-(2-methylphenyl)piperidin-4-yl]-1,4-diazepan-1-yl}propan-1-one
methyl 5-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(oxolan-2-ylmethyl)-N-({4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)furan-2-carboxamide
5,6-dimethyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}thieno[2,3-d]pyrimidin-4-amine
5-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]-1-(butan-2-yl)-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
methyl N-{2-[(3S,4R)-3-cyclopropaneamido-4-(4-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl}carbamate
1-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-3-yl}-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
2-[(2S)-2-aminohexanoyl]-N-(5-methyl-1,2-oxazol-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(3R,4S)-4-cyclopropyl-1-[4-(piperidine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-amine
2-(3,4-dichlorophenyl)-4-(3-methoxypyridine-2-carbonyl)morpholine
3,4-dimethoxy-N-[3-(1,3-thiazol-4-yl)phenyl]benzamide
3-(4-hydroxyphenyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
2-[(2,1,3-benzoxadiazol-5-ylmethyl)amino]-N-[(2-methoxyphenyl)methyl]acetamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]propane-1-sulfonamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrimidin-2-amine
2-(3-methyl-1H-pyrazol-1-yl)-N-{[6-methyl-2-(2-methylphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
3-(1-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzoyl}piperidin-3-yl)propan-1-ol
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-5-(5-methylfuran-2-yl)-1,2,4-triazin-3-amine
N,N-dimethyl-4-(4-{[2-(pyridin-3-yloxy)ethyl]amino}piperidin-1-yl)benzamide
2-{4-[(3-chloro-4,5-dimethoxyphenyl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
1-cyclopentanecarbonyl-3-propylpiperidine-3-carboxylic acid
methyl({[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-N-(1H-pyrazol-3-ylmethyl)piperidin-4-amine
(2S)-2-({[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl}amino)propanamide
5-{[(2-fluorophenyl)methyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)(2-methoxyethyl)(pyridin-3-ylmethyl)amine
3-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}benzamide
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-(thiophen-3-ylmethyl)propanamide
14-(7-methoxy-2H-1,3-benzodioxol-5-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-cyclopropyl-1-(2-{1-[2-(4-methoxyphenoxy)acetyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
N3-cyclohexyl-1-cyclopropyl-4-oxo-N5-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide