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(1s,4s)-4-hydroxy-N-(isoquinolin-5-ylmethyl)-N-methylcyclohexane-1-carboxamide
2-(dimethylamino)-N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-2-(4-fluorophenyl)acetamide
(3R)-N-(2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(4aS,7aR)-1-(1-benzofuran-5-ylmethyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-benzyl-N-methyl-3-[1-(2-oxo-2-phenylacetyl)piperidin-4-yl]propanamide
2-{[4-(2,4-dimethoxypyrimidin-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
N-[2-(4-ethylphenoxy)ethyl]-N,3-dimethylpyridine-2-carboxamide
2-{4-[3-(piperidine-1-carbonyl)pyridin-2-yl]phenoxy}acetic acid
3-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]urea
1-[(diethylcarbamoyl)methyl]-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-{[ethyl(methyl)amino]methyl}-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
3-[2-(2,3-difluorophenyl)-1H-imidazol-1-yl]-4-hydroxybenzonitrile
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-chloro-2-methylphenyl)urea
N-[3-({[(1R,2R)-2-hydroxycyclohexyl](propyl)carbamoyl}amino)phenyl]-N-methylacetamide
2-methyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-6-(piperidin-4-yl)pyrimidin-4-amine
ethyl 3-[5-(2,3-dimethoxyphenyl)-4-phenyl-1H-imidazol-1-yl]propanoate
2-cyclopentyl-N-[(4-methoxypyridin-2-yl)methyl]-2-phenylacetamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
6,7-dimethoxy-2-[1-(thian-4-yl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
4-(4-ethoxy-3-methylphenyl)-4-oxo-N-[3-(pyridin-4-yl)propyl]butanamide
N-cyclopropyl-N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-2-(thiophen-3-yl)acetamide
2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]acetamide
4-{2-[(4-benzyl-5-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}morpholine
5-[2-(benzylamino)ethyl]-1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
3-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}ethan-1-one
(3-methoxypropyl)({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
2-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-(thiophen-3-ylmethyl)acetamide
2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(phenoxymethyl)-1H-1,2,4-triazol-3-yl]acetamide
N-[(3-hydroxypyrrolidin-3-yl)methyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-[(2,2-dimethyloxan-4-yl)methyl]-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
2-(adamantan-1-yl)-5-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-(naphthalen-1-ylmethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-ethoxyfuran-2-carboxamide
1-(4-methoxyphenyl)-4-[2-(pyrrolidin-1-yl)propanoyl]piperazin-2-one
1-[(2-chlorophenyl)methyl]-N-methyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-{[ethyl(oxolan-2-ylmethyl)amino]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
N-(2-{3-[hydroxy(phenyl)methyl]-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl}ethyl)acetamide
1-amino-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)cyclobutane-1-carboxamide
N-benzyl-N,1-dimethyl-5-{[2-(methylsulfanyl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3S,4R)-1-(1H-indole-5-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-4-(2-oxopyrrolidin-1-yl)benzamide
(2R,3R,6R)-3-(4-fluorophenyl)-5-(1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]methyl}-5,8-dimethylquinolin-4-ol
N-[2-(3,4-dimethoxyphenyl)propan-2-yl]-1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
(3R,4R)-1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
9-(5-chloro-3-fluoropyridin-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol