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{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[4-(morpholin-4-yl)butyl]amine
1-{4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butanoyl}-1,4-diazepan-5-one
4-ethyl-3-(piperidin-3-yl)-1-(quinolin-8-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[(2-methylpropyl)amino]methyl}piperidin-2-one
9-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
9-(2-methoxyethyl)-1-methyl-4-(9H-purin-6-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
[1-(dimethyl-1,3-thiazol-4-yl)ethyl]({[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl})methylamine
{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl})amine
N-[2-(methylamino)ethyl]-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
[(1S)-1-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethyl]dipropylamine
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)benzamide
1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-(oxan-4-ylmethyl)piperidin-4-amine
(2-chloro-6-fluorophenyl)(4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
1-[1'-(2-hydroxy-5-methoxybenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
3-(2-ethylbutyl)-8-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{3-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]adamantan-1-yl}(methylsulfanyl)formamide
1-[1-(morpholine-4-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
1-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
4-{3-cyclopropyl-1-[(4-ethylphenyl)methyl]-1H-1,2,4-triazol-5-yl}-N-methyl-1,3-thiazol-2-amine
9-(2,5-dimethylfuran-3-carbonyl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
5-cyclopropanecarbonyl-1'-{[3-(methylsulfanyl)phenyl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine-4-carbonitrile
N-methyl-N-[3-(4-methylphenoxy)propyl]-3-(piperidin-3-yl)benzamide
3-{2-[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
N-ethyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(pentan-3-yl)-1,3-oxazole-4-carboxamide
3-methyl-5-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-pyrazole
2-{1-[1-(benzenesulfonyl)cyclopropanecarbonyl]azetidin-3-yl}pyridine
1-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-(1H-imidazol-4-yl)-1H-imidazole
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-(2-hydroxyethyl)-N-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}piperidine-4-carboxamide
2-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrazine
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(4-chloro-1H-pyrazol-1-yl)propan-1-one
1-tert-butyl-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
1-{6-[2-(trifluoromethyl)morpholin-4-yl]pyrimidin-4-yl}piperidin-4-ol
(3S,5S,9R)-5-{[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]amino}-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
1-{furo[3,2-c]pyridin-4-yl}-4-(2-phenylethyl)piperidine-4-carboxylic acid
2-(4-fluorophenyl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidine
8-[(4-methoxyphenyl)methyl]-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
[4-(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)morpholin-3-yl]methanol
ethyl 1-(3,5-dimethylfuran-2-carbonyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
(2S,4S)-1-cyclopentyl-N-ethyl-4-[2-(2-methylphenyl)acetamido]pyrrolidine-2-carboxamide
3-{1-[(3-chloro-4-hydroxyphenyl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-[(1S,2R)-2-carbamoylcyclopentyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
3-(4-fluorophenyl)-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazin-2-one
1-methyl-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine