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2-(2-methoxyethyl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-benzoxazole-6-carboxamide
2-(4-{[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}phenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
2-(pyridin-4-yl)-N-[2-(thiophen-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N3-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N5-[2-(propan-2-yloxy)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
diethyl({3-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
N-[(2R,3R)-1'-(3-chlorothiophene-2-carbonyl)-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
(4aS,8aR)-6-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
N-(2-methoxyethyl)-6-[4-(3-methoxypropyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-cyclopentyl-1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-(4-hydroxyphenyl)-1-(4-methyl-1,4-diazepan-1-yl)-2-phenylpropan-1-one
2-(4-{1,4-diazabicyclo[3.2.2]nonan-4-ylmethyl}phenyl)-6-(pyridin-2-yl)-3,4-dihydropyrimidin-4-one
N-methyl-N-(3-oxo-3-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}propyl)methanesulfonamide
2-{4-[6-(dimethylamino)pyrimidin-4-yl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-(dimethylamino)-N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(4-methylphenyl)acetamide
(4S,6R)-6-methyl-N-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}-2-sulfanylidene-1,3-diazinane-4-carboxamide
1-[cyclohexyl(methyl)amino]-3-{4-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)methyl]-2-methoxyphenoxy}propan-2-ol
1-benzyl-N,2-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carboxamide
2-(methoxymethyl)-6-methyl-1-(naphthalen-1-ylmethyl)-3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(3,5-difluoro-4-methoxyphenyl)methyl](methyl)[(3-methylpyridin-2-yl)methyl]amine
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)(methyl)[(5-methylfuran-2-yl)methyl]amine
4-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
(4aS,8aS)-2-(pyrimidin-2-yl)-decahydro-2,7-naphthyridin-4a-ol
(2R,4R)-N-[(5-chloro-2-ethoxyphenyl)methyl]-4-hydroxy-N-methylpyrrolidine-2-carboxamide
4-fluoro-2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
8-cyclopropanecarbonyl-2-(pyridine-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
3-(dimethyl-1,2-oxazol-4-yl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
(1S,6R)-3-methyl-N-[4-(morpholine-4-carbonyl)phenyl]-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}oxolane-2-carboxamide
1-ethyl-1-(oxan-2-ylmethyl)-3-(3-sulfamoylphenyl)urea
N-[4-({methyl[1-(1,2-oxazol-3-yl)ethyl]carbamoyl}methoxy)phenyl]propanamide
4-{[1-(pyridin-2-yl)propyl]amino}pyrimidine-5-carboxylic acid
6-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]piperazin-2-one
N-[(3S)-2-oxoazepan-3-yl]-4-[4-({[3-(trifluoromethyl)phenyl]methyl}amino)piperidin-1-yl]benzamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
2-{4-[(2,6-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-(dimethylamino)propan-2-ol
N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-2-propyl-1,3-thiazole-4-carboxamide
3-(2-methylpropyl)-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-1,2-oxazole-5-carboxamide
N-{2-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]ethyl}-5-methylpyrimidin-2-amine
2-(3-chloro-4-hydroxyphenyl)-1-[4-(dimethylamino)azepan-1-yl]ethan-1-one
{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amine
N-[(3S,4R)-1-(3-cyano-4,6-dimethylpyridin-2-yl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-fluoro-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methylbenzamide
N-(1-benzothiophen-2-ylmethyl)-1-ethyl-N-methyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-N-methyloxolan-3-amine
3-({[3-(dimethylamino)propyl](methyl)amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one