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N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
methyl({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})[1-(1,3-thiazol-2-yl)ethyl]amine
(3aR,6aR)-2-cyclopropanecarbonyl-5-(1,3-thiazol-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[5-(2-propyl-1,3-thiazole-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
2-(3-methyl-1H-pyrazol-1-yl)-1-(4-{4-[(methylamino)methyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)ethan-1-one
3-hexyl-8-[2-(1H-1,2,4-triazol-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2,5-dimethoxyphenyl)-N'-[(3S)-2-oxoazepan-3-yl]propanediamide
3-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
2-(4-chloro-3-methylbenzoyl)-octahydropyrrolo[1,2-a]piperazine
1-(4,5-dimethyl-1H-1,3-benzodiazol-6-yl)-3-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}urea
N-[(4-phenyloxan-4-yl)methyl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
4-[(6-cyclopropylpyrimidin-4-yl)amino]-N-ethylpiperidine-1-carboxamide
N5-cyclopropyl-N6-[2-(diethylamino)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(oxolan-3-ylmethyl)piperidine-4-carboxylic acid
3-{1,6-dimethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-5-(2,6-dimethylphenoxymethyl)-1,2-oxazole
1-{2-[1-(2,5-dimethoxybenzoyl)piperidin-2-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
methyl 2-[butyl(methyl)sulfamoyl]-6-[(4-ethoxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-hydroxy-2-(phenoxymethyl)pyrimidine-5-carboxamide
1-[3-(thiophene-2-carbonyl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-sulfamoylbenzamide
N-({7-[(2E)-3-(2,3-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)acetamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
4-{6-[4-(pyridin-2-yl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}thiomorpholine
N-(2-hydroxyethyl)-6-(4-methoxyphenyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[(2,6-dimethoxyphenyl)methyl]-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-benzyl-N-ethyl-3-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
ethyl 2-(2-{[5-(phenoxymethyl)-1,2-oxazol-3-yl]formamido}ethyl)-1,3-thiazole-4-carboxylate
N-(2-{[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]amino}ethyl)pyridine-4-carboxamide
N-[2-(3-fluorophenyl)ethyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
[(2-ethylpyrimidin-5-yl)methyl](methyl)(pyrazin-2-ylmethyl)amine
(1S,3R)-N1-[(5-fluoro-1H-indol-2-yl)methyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-methoxy-N-{[1-(4,4,4-trifluorobutanoyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
1-ethyl-3-methyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]piperidine-3-carboxamide
1-[4-(benzenesulfonyl)piperazin-1-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
(4aR,8aS)-1-butyl-6-{[5-(3-chlorophenyl)furan-2-yl]methyl}-decahydro-1,6-naphthyridin-2-one
(3S,4S)-1-(3-cyano-6-methylpyridin-2-yl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
5-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
N-{2-cyclobutyl-1-methyl-7-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
[(2-phenoxypyridin-3-yl)methyl]({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl})amine
2-(2H-1,3-benzodioxol-5-yl)-N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-4-ylmethyl)acetamide
3-methoxy-1-{2-oxo-2-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]ethyl}-1,2-dihydropyridin-2-one
3-methyl-6-[5-(1-propoxyethyl)-1,2,4-oxadiazol-3-yl]pyridazine
2-{[3-(2-hydroxyethyl)-4-(2-phenylethyl)piperazin-1-yl]methyl}quinolin-4-ol
1-(3-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-oxopropyl)azepan-2-one
1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}acetamide
(4aS,8aR)-1-(2-propoxyethyl)-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
2-ethoxy-6-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}phenol
4-(1-{1-[2-(difluoromethoxy)benzoyl]piperidin-4-yl}ethyl)morpholine