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1-ethyl-5-[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-[1-(2,4,5-trimethylphenyl)-1H-pyrazol-4-yl]ethan-1-ol
[(3R,4R)-1-(5-propyl-1,2-oxazole-3-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-(2-ethyl-4-methyl-1,3-oxazol-5-yl)-3-(2-methoxyethyl)-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazole
(3aS,6aS)-2-[3-(methylsulfanyl)propyl]-5-(thiophen-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{5-[(3-chlorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
N-[(2-fluorophenyl)methyl]-2-[2-(pyridin-2-yl)piperidin-1-yl]acetamide
1-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]piperidine-4-carbonitrile
N-(2-methyl-4-{[1-(1H-1,2,4-triazol-5-yl)ethyl]carbamoyl}phenyl)furan-2-carboxamide
1-(4-methyl-1,4-diazepan-1-yl)-2-[(1-methyl-1H-indol-3-yl)sulfanyl]ethan-1-one
6-oxo-N-[2-(pyridin-3-yloxy)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
4-(5-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
(1S,5R)-3-cyclobutanecarbonyl-6-[3-(difluoromethoxy)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
1-(5-ethyl-1,2,4-oxadiazol-3-yl)-3-(3-methoxypropyl)piperidine
1-[(4-methoxyphenyl)methyl]-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-one
2-[2-({3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)phenoxy]ethan-1-ol
3-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-(3-methyl-1-propyl-1H-pyrazol-5-yl)urea
N-[1-({[(4-fluorophenyl)methyl](methyl)carbamoyl}methyl)-1H-pyrazol-4-yl]-4-oxo-4-phenylbutanamide
3-cyclohexyl-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-1,2-oxazole
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-8-(quinoxalin-2-yl)-1,8-diazaspiro[4.5]decane
4-({5-[3-(2-fluorophenyl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
4-(3-methoxypropyl)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylthiophene-2-carboxamide
methyl (2S,4R)-1-[(2,5-dimethylphenyl)methyl]-4-[2-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
N-[1-(furan-2-yl)ethyl]-9-methoxy-3-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-1-(propan-2-yl)piperidine-4-carboxamide
2-[1-(1-benzoxepine-4-carbonyl)pyrrolidin-2-yl]-6-methyl-1H-1,3-benzodiazole
(1R,2R)-2-{ethyl[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amino}cyclohexan-1-ol
5-{[4-(1H-imidazol-2-yl)piperidin-1-yl]methyl}-N-(propan-2-yl)pyrimidin-2-amine
{1-[2-({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)ethyl]piperidin-2-yl}methanol
N-[(2R,3R)-1'-[2-(2H-indazol-2-yl)acetyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxyacetamide
5-(3-acetylphenoxymethyl)-N-[3-(propan-2-yloxy)propyl]-1,2-oxazole-3-carboxamide
3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}propanamide
N-benzyl-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
2-[(4-fluorophenyl)methyl]-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}morpholine
3-(2-phenoxyethyl)-8-[3-(pyrrolidin-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-{1-[2-(2-fluorophenyl)acetyl]piperidin-4-yl}-5-[(4-fluorophenyl)methyl]-3-(oxolan-3-yl)imidazolidine-2,4-dione
2-oxo-6-phenyl-N-propyl-N-(thiophen-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-methyl-5-{[3-(2-methylphenyl)phenyl]methyl}-N-[3-(morpholin-4-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[2-({7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)ethyl]-1,3-thiazol-2-amine
1-(dimethyl-1,2-oxazole-4-carbonyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine
2-methyl-5-(3-{[(pentan-3-yl)amino]methyl}pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
1-[1-(propan-2-yl)piperidin-4-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-2-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]propanamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyridine-4-carboxamide
4-{[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]methyl}-1-ethyl-1H-pyrrole-2-carbonitrile
[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](furan-3-ylmethyl)methylamine
N-[4-(propylsulfanyl)phenyl]-3-(pyridin-3-yl)azetidine-1-carboxamide
2-(3-fluoro-4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-(oxolan-2-ylmethyl)benzamide