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1-[4-(furan-2-ylmethoxy)phenyl]-3-methyl-3-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}urea
3-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3H,4H-pyrido[2,3-d]pyrimidin-4-one
(4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholin-2-yl)methanamine
(1s,5s)-3,7-dimethyl-10-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-3,7,10-triazatricyclo[3.3.3.01,5]undecane
N-(1-benzylpiperidin-3-yl)-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-(2-{3-[2-(2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]morpholin-4-yl}-2-oxoethyl)imidazolidine-2,4-dione
4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]piperazin-2-one
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
N-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-N-methyloxan-4-amine
N1,N1-dimethyl-N3-(2-methylpropyl)-N3-(pyridin-2-ylmethyl)piperidine-1,3-dicarboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
2-(1-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)pyridine
2-cyclohexyl-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
4-[(5-{1-[2-(ethylsulfanyl)ethyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
1-(2-methyl-1-benzofuran-7-carbonyl)-4-[(2-methylphenyl)methyl]piperazine
7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-3-methylimidazolidin-2-one
N-[2-(7-{[4-(2-methylpropyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]pyridine-3-carboxamide
3,5-dimethoxy-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}benzamide
2-[4-(2-cyclohexyl-1,3-benzoxazole-6-carbonyl)piperazin-1-yl]-N-(propan-2-yl)acetamide
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
1-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-4-(oxolane-2-carbonyl)piperazine
2-(2-methoxy-4-methylphenoxymethyl)-N-[(1R,2S)-2-phenylcyclopropyl]-1,3-oxazole-4-carboxamide
5-chloro-4-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}-2-methoxyphenol
5-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
1-[(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
4-(4-chlorophenoxy)-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-4-carboxamide
2-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]benzoic acid
2-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-2-yl}-1H-1,3-benzodiazole
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[6-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methanol
4-methyl-N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}-1,2,3-thiadiazole-5-carboxamide
5-[6-(piperidin-1-yl)pyrimidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-(4-methoxyphenyl)-1,2,4-triazin-3-amine
2-(dimethylamino)-4-methyl-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)pyrimidine-5-carboxamide
2-[(4aR,8aR)-4a-hydroxy-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-2-yl]-6-methylpyridine-3-carbonitrile
5-[1-(2-methoxyacetyl)pyrrolidin-2-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]thiophene-2-carboxamide
1-(4-methoxyphenyl)-3-methyl-4-(pyridazine-3-carbonyl)piperazin-2-one
N-[(5-methylpyrazin-2-yl)methyl]-1-(9H-purin-6-yl)piperidin-4-amine
{9-[4-(methylamino)pyrimidin-2-yl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
1-[(dimethyl-1,3-thiazol-5-yl)methyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
(3R,4R)-1-(furan-3-ylmethyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3,5-dimethyl-1,2-oxazole-4-sulfonamide
2-{[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-(3-hydroxy-1-phenylpropyl)-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[4-(4-{[2-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)phenyl]benzenesulfonamide
7-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}-2,3-dimethyl-1H-indole
4-{1-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]-2-methylpropan-2-yl}morpholine
N-({7-[(3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
9-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-6-oxa-9-azaspiro[4.5]decane